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(2R,6R)-4-[(3-methylpyridin-4-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(morpholin-4-yl)propanamide
1-[2-(azetidin-1-ylmethyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N5-(butan-2-yl)-1-cyclopentyl-N3-ethyl-N3-(2-methylprop-2-en-1-yl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
methyl 3-({2-[(1-acetylpiperidin-4-yl)oxy]-5-chlorophenyl}formamido)propanoate
1-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,2-dihydroquinolin-2-one
N,N-dimethyl-2-[({thieno[2,3-d]pyrimidin-4-yl}amino)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-methyl-3-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}-N-(thiophen-3-ylmethyl)benzamide
8-(4,6-dimethylpyridine-3-carbonyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-3-(piperidin-4-ylmethyl)benzamide
1-benzyl-4-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
N-({2-[4-(3-chlorophenyl)piperazin-1-yl]-7-fluoroquinolin-3-yl}methyl)cyclopropanamine
1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]-4-(pyridin-2-yl)piperidin-4-ol
{1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}(thiophen-2-yl)methanol
7-[(2S)-2-amino-3,3-dimethylbutanoyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-{[1-(2,1-benzoxazole-3-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
(2S,4R)-4-amino-1-[2-(4-amino-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-N-ethylpyrrolidine-2-carboxamide
4-[4-(4-methyl-1,3-thiazole-5-carbonyl)piperazin-1-yl]quinazoline
1-ethyl-3-{2-[4-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
N-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}-1-(2-fluorophenyl)piperidin-4-amine
3,5-dichloro-N,4-dimethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]benzamide
N-[(3R,4S)-1-acetyl-4-propylpyrrolidin-3-yl]-2-(5,5-dimethyl-2,4-dioxoimidazolidin-1-yl)acetamide
(3R,5S)-1-benzyl-5-(3-fluorophenoxymethyl)-N-[3-(morpholin-4-yl)propyl]piperidine-3-carboxamide
1-ethyl-N-(furan-3-ylmethyl)-N-methyl-5-[(prop-2-en-1-yl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-ethyl-3-methyl-N-[2-(4-sulfamoylphenyl)ethyl]piperidine-3-carboxamide
methyl 1-{9-methoxy-3-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
1-phenyl-N-{[7-(pyrimidin-2-yl)-1H,2H-naphtho[2,1-b]furan-2-yl]methyl}cyclopropane-1-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-5-phenyl-1,2-oxazole-3-carboxamide
1-(pyridin-2-ylmethyl)-4-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazine
1-[(1-ethyl-1H-indol-4-yl)methyl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
N-[(1-ethylpyrrolidin-2-yl)methyl]-5-methoxy-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}furan-2-carboxamide
N-({4-[(2-chloroprop-2-en-1-yl)oxy]phenyl}methyl)-2-methoxy-N-(pyridin-3-ylmethyl)benzamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-(1-methyl-1H-indol-3-yl)-N-(pyridin-3-ylmethyl)acetamide
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-2-oxo-2H-chromene-3-carboxamide
3-(2-amino-4-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-6-methylpyrimidin-5-yl)propanoic acid
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[3-(trifluoromethyl)benzoyl]piperidine
5-[3-(methylsulfanyl)phenyl]-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
3-[3-({[(1-methyl-1H-imidazol-2-yl)methyl](propyl)amino}methyl)-1H-indol-1-yl]propanamide
3-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-4-yl]-1-(pyrrolidin-1-yl)propan-1-one
2-({[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
1-(3-{[({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
N-methyl-2-{2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}ethane-1-sulfonamide
ethyl 1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-4-carboxylate
(2H-1,3-benzodioxol-5-ylmethyl)({[3-(1H-pyrazol-4-yl)phenyl]methyl})amine
2-{1-cyclopentyl-4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
{1-ethyl-5-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
3-(3-methoxyphenyl)-4-(propan-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
6-{[3-(2-hydroxyethoxy)phenyl]methyl}-N-(2-methoxyphenyl)-6-azaspiro[2.5]octane-1-carboxamide