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4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(2-methylpropanesulfonyl)ethyl]benzamide
(2S,4R)-4-amino-N-ethyl-1-[3-(1H-pyrazol-4-yl)benzoyl]pyrrolidine-2-carboxamide
3-(2-chlorophenyl)-1-(4-fluorophenyl)-4-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-1H-pyrazole
2,3,5,6-tetramethyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
2-methoxy-5-({2-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)benzoic acid
3-ethyl-5-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1,2-oxazole-4-carboxamide
N-({7-[2-(4-methoxyphenyl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-4-carboxamide
4-(1,3-benzothiazol-2-yl)-2-({[2-(3-fluorophenyl)ethyl]amino}methyl)phenol
1-{2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethyl}-1H-imidazole
1-methyl-1'-(5-propyl-1,2,4-oxadiazol-3-yl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
{1-[3-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]piperidin-2-yl}methanol
2-cyclopropyl-6-[4-(furan-2-carbonyl)-1,4-diazepane-1-carbonyl]-1,3-benzoxazole
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-3-(1-methylpiperidin-2-yl)propanamide
1-{3-[(4-fluorophenyl)methyl]-1,2-oxazole-5-carbonyl}-3-(3-methylphenyl)piperidine
N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]furan-3-carboxamide
4-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}-5-(hydroxymethyl)-2-methylpyridin-3-ol
4-[4-(ethanesulfonyl)piperazin-1-yl]-6-(morpholin-4-yl)pyrimidin-2-amine
1-(4-methyl-1,4-diazepane-1-carbonyl)-6-[(4-phenylphenyl)methyl]-6-azaspiro[2.5]octane
4-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-methyl-4-{5-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]furan-2-yl}but-3-yn-2-ol
2-(2,4-difluorophenyl)-2-{2-[1-(propan-2-yl)piperidin-4-yl]acetamido}acetic acid
1-ethyl-5-[methyl({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)-1H-imidazole-2-carboxamide
6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-[2-(methylsulfanyl)acetyl]-1,4-diazepan-2-one
N-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-N-methylthian-4-amine
3-(1,2-oxazinan-2-yl)-N-(2-propoxyethyl)propanamide
4-phenyl-3-(piperidin-4-yl)-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(2,3-dihydro-1H-inden-2-yl)-8-{[5-(hydroxymethyl)furan-2-yl]methyl}-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N'-[3-(azepan-1-yl)propyl]-N-(2,3-dimethylphenyl)-N'-methylpropanediamide
8-[(3-methoxyphenyl)methyl]-1-(2-phenylethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-({4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)acetic acid
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}morpholine-2-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine-2-carboxamide
N1,N1,2,2,3-pentamethyl-N3-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}cyclopentane-1,3-dicarboxamide
N-cyclopropyl-6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-N-propyl-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)acetamide
2-[(3-methoxyphenyl)amino]-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)butanamide
N-methyl-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]-N-[(5-propyl-1H-pyrazol-3-yl)methyl]acetamide
6-{1-[(8-methoxy-2H-chromen-3-yl)methyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
2-hydroxy-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}acetamide
N-methyl-N-{1-[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]pyrrolidin-3-yl}acetamide
2-[1-cyclopentyl-3-(2-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
{3-[(4-fluorophenyl)methyl]-1-[(2-methoxynaphthalen-1-yl)methyl]piperidin-3-yl}methanol
4-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]azepane
6-(cyclohex-3-ene-1-carbonyl)-3-(2,4-difluorophenyl)-1-(pyridin-2-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-{2-methyl-1-[7-(naphthalen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]propyl}methanesulfonamide
N-cyclopropyl-N-{[4-methoxy-3-(pyridin-4-ylmethoxy)phenyl]methyl}-4-phenylbenzamide
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-2-[(3-methoxyphenyl)amino]butanamide
5-ethyl-2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide