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1-(4-fluorophenyl)-4-[7-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butane-1,4-dione
ethyl 1-{3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperidine-3-carboxylate
N-[3-(3-fluorophenyl)phenyl]-1-[(5-methylfuran-2-yl)methyl]piperidine-4-carboxamide
[(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)(1,3-thiazol-2-ylmethyl)amine
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(3,3,4,4-tetrafluorobutyl)piperidine
2-(2-chloro-6-fluorophenyl)-1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]ethan-1-one
methyl 4-({2-[(4-methoxyphenyl)methyl]-1,3-benzoxazol-6-yl}formamido)butanoate
N-{1-[4-(3-chlorophenyl)-5-[(cyclohexylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}-2-(1-methyl-1H-pyrrol-3-yl)acetamide
N-(2-methyl-1,3-benzothiazol-6-yl)-2-propyl-2,5-dihydro-1H-pyrrole-1-carboxamide
2-{[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]methyl}pyridine
1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
4-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]benzoic acid
5-{1-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-1H-imidazol-2-yl}-N,N-dimethylpyrimidin-2-amine
2-amino-1-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]ethan-1-one
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-[(3-fluorophenyl)methyl]-N-methyl-4,5-dihydro-1,2-oxazole-5-carboxamide
N-[3-(2-ethoxyphenyl)propyl]-5,6-dimethylpyridine-3-carboxamide
3-[4-(methylsulfanyl)benzoyl]-1-(1H-pyrazol-3-ylmethyl)piperidine
2-{5-[4-(piperidin-1-ylmethyl)benzoyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-3-(2,5-dioxoimidazolidin-4-yl)-N-methylpropanamide
3-methyl-7-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
methyl 4-(4-{[(2S)-4-ethyl-2-methyl-3-oxopiperazin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
7-(2-methylphenyl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-1-ethyl-1H-pyrazole
2-[(2,3-dimethoxyphenyl)methyl]-4-[4-(2-methylbenzoyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
methyl 5-(3-{[3-(1H-indol-2-yl)phenyl]carbamoyl}piperidin-1-yl)-5-oxopentanoate
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-2-(propan-2-yl)-1,3-thiazole-4-carboxamide
{1-[(3,4-dimethoxypyridin-2-yl)methyl]-3-(3-methylbut-2-en-1-yl)piperidin-3-yl}methanol
3-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]azetidin-3-yl}pyridine
N-cyclopropyl-3-fluoro-N-{[4-methoxy-3-(pyridin-4-ylmethoxy)phenyl]methyl}benzamide
2-amino-3-ethyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-cyclohexyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1H-pyrazole-4-carboxamide
1-(2-aminoethyl)-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
methyl 3-({1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-1H-1,3-benzodiazol-7-yl}formamido)propanoate
1-(2,1,3-benzoxadiazol-4-ylmethyl)-N-[3-(3-fluorophenyl)phenyl]piperidine-4-carboxamide
2-propyl-8-(9H-purin-6-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-(1-ethyl-1H-imidazol-2-yl)-1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]piperidine
3-phenoxy-N-{1-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
N-[cyclopropyl(pyridin-2-yl)methyl]-N,1,3,7-tetramethyl-1H-indole-2-carboxamide
4-benzyl-1-methyl-3-{1-[(2-methylpyrimidin-5-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-[4-(piperidine-1-carbonyl)piperidin-1-yl]ethan-1-one
1-(pyridin-3-ylmethyl)-4-[(1s,4s)-4-aminocyclohexyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-4-(oxan-4-yl)piperazine
1-(cyclohexylmethyl)-N-ethyl-4-oxo-5-[4-(thiophene-2-carbonyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
N-[2-(4-methoxybenzenesulfonamido)ethyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
1-(3-cyanophenyl)-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
3-[2-(azepan-1-yl)-2-oxoethyl]-4-[(3,5-dimethoxyphenyl)methyl]piperazin-2-one
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amine
(3S,4S)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-(2-amino-4-methyl-1,3-thiazol-5-yl)-1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]ethan-1-one