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methyl 3-{[1-(cyclopropylmethyl)-5-[(2-methyl-1H-indol-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-6-(2-methylpiperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
N-methyl-2-[4-(4-methyl-1,4-diazepan-1-yl)-6-oxo-1,6-dihydropyridazin-1-yl]-N-(1,3-thiazol-2-ylmethyl)acetamide
1-(2-ethoxyphenyl)-4-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazine
4-[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
4-({1-[2-(1H-pyrazol-1-yl)benzoyl]piperidin-2-yl}methyl)morpholine
5-cyclohexaneamido-N-[(4-fluorophenyl)methyl]-1-(2-methoxyethyl)-N-methyl-1H-1,3-benzodiazole-7-carboxamide
(1S,5R)-6-[(1R,5S,6R)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-3-benzoyl-3,6-diazabicyclo[3.2.2]nonane
3-(1H-1,3-benzodiazol-2-yl)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]propanamide
2-{[6-(2-aminoethyl)pyrimidin-4-yl]amino}-N-tert-butylacetamide
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]propanamide
3-(2-phenylethyl)-5-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-yl}-1H-1,2,4-triazole
5-methyl-4-{[1-(3-methylbutanoyl)piperidin-4-yl]amino}thieno[2,3-d]pyrimidine-6-carboxylic acid
2-chloro-5-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)pyridine
5-(2-methoxyacetamido)-1-methyl-2-(pyridin-4-yl)-N-[1-(thiophen-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-{[3-(1H-pyrazol-1-yl)azetidin-1-yl]methyl}piperidin-2-one
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-2-(pyridin-2-yl)acetamide
(1R,3S)-7-(5-chloro-2-fluorobenzoyl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-{[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}acetamide
3-{1-[(4-methoxynaphthalen-1-yl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
(2S,4S)-4-({[4-(benzyloxy)phenyl]methyl}amino)-1-[(4-chlorophenyl)methyl]-N-ethylpyrrolidine-2-carboxamide
2-[2-(2,3-dihydro-1-benzofuran-5-yl)-1H-1,3-benzodiazol-1-yl]ethan-1-ol
3-{[(1-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}piperidin-3-yl)oxy]methyl}pyridine
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-methylurea
1-(2-methyloxane-2-carbonyl)-4-(4-methylphenoxy)piperidine
1-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)benzoyl]-4-(3-methylpyridin-2-yl)piperazine
methyl 7-oxo-3-(pyridine-4-carbonyl)-9-(thiophen-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-(1H-imidazol-2-yl)-1-[1-(oxolane-2-carbonyl)piperidine-4-carbonyl]piperidine
2-{4-[4-(2,3-dihydro-1H-isoindole-2-carbonyl)-6-fluoroquinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol
5-(2-cyclopentylacetamido)-1-methyl-2-(oxolan-2-yl)-N-(pyridin-4-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
5-[2,2-bis(prop-2-en-1-yl)piperidine-1-carbonyl]-1-(3-phenylpropyl)piperidin-2-one
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-[3-(piperidin-1-yl)propyl]propanamide
5-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}-2,1,3-benzoxadiazole
3-{1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-3-yl}benzoic acid
6-methoxy-2-oxo-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-[3-(cyclopropylmethyl)-5-[2-(1H-pyrazol-1-yl)phenyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
4-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
3-[4-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)-1H-pyrazol-1-yl]propanoic acid
8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
3-benzyl-4-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperazin-2-one
1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidine-1-carbonyl}cyclopropan-1-amine
3-(2-{[(1,5-dimethyl-1H-indazol-3-yl)methyl]amino}propyl)-3,4-dihydroquinazolin-4-one
3-({methyl[(3-phenyl-1,2-oxazol-5-yl)methyl]amino}methyl)quinolin-7-ol
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
1-(4-methoxyphenyl)-2,2-dimethyl-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
4-(1H-pyrazol-4-yl)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
(1R,9S)-11-(2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetyl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one