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N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-5-phenyl-1H-pyrazole-3-carboxamide
(2E)-1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-3-(1H-imidazol-4-yl)prop-2-en-1-one
1-[(2,3-difluorophenyl)methyl]-4-[1-(1-methylcyclopropanecarbonyl)pyrrolidin-3-yl]piperidine
9-{2-methyl-2,7-diazaspiro[4.5]decan-7-yl}-3-azaspiro[5.5]undecane
ethyl 5-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
8-(4-aminopyrimidin-2-yl)-2-cyclopropanecarbonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(4-{4-[(1,2-oxazol-3-ylmethyl)amino]piperidin-1-yl}phenyl)-5-phenylpentanamide
5-[1-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)piperidin-4-yl]-5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
4-(5-methylpyridin-2-yl)-1-(2-methylpyridine-3-carbonyl)piperidin-4-ol
1-methyl-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-1H-indole-3-carboxamide
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
2-(2-hydroxyethyl)-8-(5-methylthiophene-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
[(2S,4R,5R)-5-(4-chlorophenyl)-1-ethyl-4-({[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]amino}methyl)-2-methylpyrrolidin-2-yl]methanol
N-methyl-2-(1-methyl-1H-pyrrol-2-yl)-2-oxo-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
2-[4-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)phenoxy]acetic acid
N-({5-methyl-2-[3-(2-methylfuran-3-amido)phenyl]-1,3-oxazol-4-yl}methyl)quinoline-2-carboxamide
3-(3-methylpiperidin-1-yl)-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-5,6-dimethylpyrimidin-4-amine
6-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-2-(pyridine-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline
(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-4-(2-phenoxyethyl)piperidin-4-yl)methanol
2-ethyl-N-({5-methyl-2-[3-(3-methylbutanamido)phenyl]-1,3-oxazol-4-yl}methyl)butanamide
N-cyclopropyl-3-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-({3-[(dimethylamino)methyl]phenyl}methyl)-N-methylpyrimidin-2-amine
5-(2,2-diethylcyclopropanecarbonyl)-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[2-(dimethylamino)-2-(furan-2-yl)ethyl]-6-ethylpyrimidin-4-amine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}butan-1-one
3-[4-hydroxy-4-(hydroxymethyl)azepane-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
N-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-methylpropyl]-6-ethylpyrimidin-4-amine
N-{1-benzyl-2-methyl-7-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl}acetamide
N-benzyl-2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
5-tert-butyl-N-[2-(dimethylamino)-3-methylbutyl]-1,3,4-oxadiazol-2-amine
1-{3-oxo-3-[3-(phenylamino)piperidin-1-yl]propyl}piperidin-2-one
1-{3-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}propan-1-one
1-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1H-indole-2-carboxamide
1-[(2-chlorophenyl)methyl]-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-1-ethylpiperidin-4-amine
4-{4-[4-(benzyloxy)piperidin-1-yl]piperidin-1-yl}-N-(pyridin-3-ylmethyl)benzamide
1-(2-methoxyethyl)-4-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carbonyl}piperazine
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-4-(1H-pyrazol-1-yl)benzamide
1-({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)-1,4-diazepan-5-one
(2S,4S)-N-[2-(dimethylamino)ethyl]-4-[(4-fluorophenyl)sulfanyl]-1-[(3-methylphenyl)methyl]pyrrolidine-2-carboxamide
5-methyl-N-[1-(pyridin-3-yl)pentyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-(5-methylhexan-2-yl)piperidin-3-amine
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
1-[(4-fluorophenyl)methyl]-N-[3-(1H-imidazol-1-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
(4aS,7aR)-4-acetyl-N-[(2-fluorophenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-3-(quinolin-5-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-({2-amino-6-[4-(4-fluorophenoxy)piperidin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
3-{1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}-N-phenylpropanamide