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N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-(methylsulfanyl)acetamide
5-[1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-4-methylpyrimidin-2-amine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(furan-3-ylmethyl)pyrrolidin-3-yl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(2-{5-methyl-4-[(2-phenoxypropanamido)methyl]-1,3-oxazol-2-yl}phenyl)pyridine-3-carboxamide
1-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]-2-(1,2-benzoxazol-3-yl)ethan-1-one
1-cycloheptyl-4-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(thiophen-3-yl)acetamide
5-{[(3,4-dimethoxyphenyl)methyl]amino}-1-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-(1H-imidazol-1-yl)-1-[3-(pyridine-2-carbonyl)piperidin-1-yl]propan-1-one
1-(3,5-dimethylphenyl)-4-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-2-one
1-[2-(3-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[3-(furan-2-yl)phenyl]-1-(1,3-thiazol-2-ylmethyl)piperidine-4-carboxamide
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-{3-[(pyridin-3-yl)amino]propyl}urea
N-[(1-ethylpiperidin-3-yl)methyl]-2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-methylacetamide
4-methyl-6-(4-{[phenyl(pyridin-4-yl)methyl]amino}piperidin-1-yl)pyrimidin-2-amine
N-(furan-2-ylmethyl)-N,1-dimethyl-5-[(3-phenylpropyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(2-{7-[(2,3,4-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1,4-diazepane
N-(2-{7-[(3-phenoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
2-(3-methyl-4-oxo-3,4-dihydroquinazoline-7-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(3-methoxyphenyl)phenyl]-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidine-4-carboxamide
(3S,4R)-1-(5-propyl-1,3,4-thiadiazol-2-yl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
6-amino-N-{1,9-dioxaspiro[5.5]undecan-4-yl}pyridine-2-carboxamide
2-{[4-(3-chlorophenyl)-5-(1-ethyl-1H-pyrazol-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-benzyl-1-[(2,3-dimethoxyphenyl)methyl]-N-methylpiperidin-3-amine
methyl (2S,4S,5R)-5-(4-chlorophenyl)-1,2-dimethyl-4-{[3-(methylsulfanyl)propyl]carbamoyl}pyrrolidine-2-carboxylate
2-(2,4-difluorophenoxy)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]acetamide
4-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]sulfonyl}-2,1,3-benzothiadiazole
2-ethyl-7-methoxy-4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-N-{2-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]phenyl}thiophene-2-carboxamide
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-[(2,4-dimethylphenyl)methyl]-1,4-diazepan-5-one
3-{1-[(3-acetylphenyl)methyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}propan-1-one
(1S,3R)-N1-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,2,N2,N3,3-pentamethylcyclopentane-1,3-dicarboxamide
1-({1-[2-hydroxy-3-(2-methylphenoxy)propanoyl]piperidin-4-yl}methyl)pyrrolidin-2-one
1-[1-(2-aminopyrimidin-4-yl)piperidin-4-yl]-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
3-(2-{2-oxa-7-azaspiro[4.5]decan-7-yl}-2-oxoethyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
1-cyclobutanecarbonyl-N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]piperidine-4-carboxamide
3-[3-(morpholin-4-yl)propyl]-1-[4-(oxolan-2-ylmethoxy)phenyl]urea
ethyl 1-[3-(naphthalen-1-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperidine-4-carboxylate
methyl({[3-({1-[4-(piperidin-1-yl)benzoyl]piperidin-3-yl}methoxy)phenyl]methyl})(quinolin-6-ylmethyl)amine
(2E)-1-{3-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-3-(pyridin-4-yl)prop-2-en-1-one
2,7,8-trimethyl-N-[(3S)-2-oxoazepan-3-yl]quinoline-4-carboxamide
3-methyl-9-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-3,9-diazaspiro[5.6]dodecane
methyl (2S)-1-(9-methoxy-7-oxo-3-{[4-(propan-2-yloxy)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl)pyrrolidine-2-carboxylate
3-(1-{imidazo[1,2-a]pyridine-6-carbonyl}pyrrolidin-2-yl)pyridine
6-methoxy-N-(3-methyl-1,2,4-thiadiazol-5-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
N-({5-[(3-cyanophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
ethyl({[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl})(pyridin-4-ylmethyl)amine
N-({7-[(2E)-3-(4-methoxyphenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)methanesulfonamide