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3-[3,5-dimethyl-1-(1H-1,2,3,4-tetrazol-5-yl)-1H-pyrazol-4-yl]-2-ethoxypyridine
N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)imidazo[1,2-a]pyrimidine-2-carboxamide
methyl 1-{2-hydroxy-3-[4-(morpholin-4-ylmethyl)phenoxy]propyl}piperidine-4-carboxylate
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl})amine
7-[(4-fluorophenyl)methyl]-2-[(6-methylpyridin-2-yl)methyl]-2,7-diazaspiro[4.5]decane
2-(2,5-dimethoxyphenyl)-5-methyl-4-(1H-pyrazol-1-ylmethyl)-1,3-oxazole
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(quinolin-5-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[(2,5-difluorophenyl)methyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
2-chloro-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}benzene-1-sulfonamide
2-{2-[2-(2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]ethyl}-5,6-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
5-amino-4-chloro-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1H-pyrazole-3-carboxamide
7-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
5-{1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]piperidin-4-yl}-3-(furan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
(2-methoxyethyl)[(4-methylphenyl)methyl](oxolan-3-ylmethyl)amine
2-[5-(1-ethyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]-3-hydroxypropanoic acid
1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-methyl-3-[1-(thiophen-2-yl)ethyl]urea
2-fluoro-N-[1-(2-oxo-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-1H-pyrazol-4-yl]benzamide
4-chloro-N-ethyl-2-methoxy-N-[(2E)-3-phenylprop-2-en-1-yl]benzamide
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carboxamide
5-chloro-3-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
5-acetyl-N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]thiophene-3-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamide
2-fluoro-N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzene-1-sulfonamide
1-[2-(dimethylamino)-4-[(3-phenylpropyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
(4aS,8aR)-6-(2-amino-4-methylpyrimidine-5-carbonyl)-1-(3-aminopropyl)-decahydro-1,6-naphthyridin-2-one
2-{1-[3-(1H-imidazol-1-yl)propyl]-1H-1,2,3-triazol-4-yl}-8-methoxyquinoline
2-amino-8-(5-chloro-2,4-dimethoxyphenyl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
4-{[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-4-ylmethyl)benzamide
6-[(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)amino]-N,N-dimethylpyridine-3-carboxamide
5-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]pyridine-2-carbonitrile
{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[2-(trifluoromethyl)phenyl]methyl}amine
5-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-5-[(3-fluorophenyl)methyl]-3-(2-methylpropyl)imidazolidine-2,4-dione
2-[1-cyclopentyl-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(dicyclopropylmethyl)-N-methylacetamide
3-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-1-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]urea
5-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}-3-(furan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
[2-(2-{[2-(4-chlorophenyl)morpholin-4-yl]methyl}phenoxy)ethyl]dimethylamine
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(2-oxo-1,2-dihydropyridin-1-yl)propanamide
7-(2-methoxy-4-methylbenzenesulfonyl)-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
8-(1,3-benzothiazol-2-ylmethyl)-3-benzyl-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{1-[(2-ethoxyphenyl)methyl]-4-[(1-ethyl-1H-imidazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[(4-fluorophenyl)methyl]-5-(4-formyl-1,4-diazepan-1-yl)-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(3-methyl-1H-pyrazol-1-yl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
1-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}pyrrolidin-2-one
5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-N-(propan-2-yl)furan-2-carboxamide
[(3R,4R)-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
1-(1-methanesulfonylpyrrolidine-2-carbonyl)-4-(2-phenylethyl)piperidine
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-phenoxybenzamide
N-ethyl-N-(4-hydroxybutyl)-3-(piperidin-3-yl)benzamide
methyl 3-(2,1,3-benzothiadiazol-5-ylmethyl)-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}urea