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N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]pyrazine-2-carboxamide
2-[(4-fluorophenyl)methyl]-4-[(6-methylpyridin-2-yl)methyl]morpholine
N-[(2-chloro-4-fluorophenyl)methyl]-2-ethyl-2H-1,2,3,4-tetrazol-5-amine
N-(2-hydroxyethyl)-1-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-[(2-methylphenyl)methyl]pyridin-2-amine
2-(2H-1,2,3-benzotriazol-2-yl)-1-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}ethan-1-one
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
4-[(3,4-dichlorophenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
2-[(2,6-dichlorophenyl)methyl]-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-hydroxypyrimidine-5-carboxamide
6-[1-(2,4-dimethylphenyl)-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]piperazin-2-one
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-[(4-propylpiperazin-1-yl)methyl]piperidin-2-one
4-[4-(5-chloro-2-methoxyphenyl)-1H-pyrazol-5-yl]pyridine
3-[2-(2,6-difluorophenyl)ethyl]-1-(prop-2-ene-1-sulfonyl)piperidine
1-{3-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
2-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-2,8-diazaspiro[4.5]decane
1-[(3-fluorophenyl)methyl]-4-[1-(2-methoxyethyl)-6-oxopiperidine-3-carbonyl]piperazin-2-one
9-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(1-benzothiophen-2-ylmethyl)-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-methylpropanamide
(2S)-N-(1-tert-butyl-4-phenyl-1H-pyrazol-5-yl)-2-(methoxymethyl)pyrrolidine-1-carboxamide
N,2-dimethyl-N-[2-(oxan-4-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
(3R,4S)-4-cyclopropyl-1-(5-ethyl-2-methylpyrimidin-4-yl)pyrrolidin-3-amine
1-methyl-1'-(thiophen-2-ylmethyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]-2,3,4-trimethoxybenzamide
2-(furan-2-yl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-oxoacetamide
1-(2-ethoxyethyl)-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
4-(3,5-dimethyl-1-benzofuran-2-yl)-3-methyl-4H,5H,6H,7H-[1,2]oxazolo[5,4-b]pyridin-6-one
4-(4-hydroxybutyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-phenylbenzamide
1-{7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-(piperidin-1-yl)ethan-1-one
4-(4-methoxyphenyl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-4-oxobutanamide
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-N,N-dimethylazepan-4-amine
5-[(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)amino]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-[(2-methylphenyl)methyl]-4-(1H-pyrrole-3-carbonyl)piperazine
N-tert-butyl-3-[2-(4-chlorophenyl)morpholin-4-yl]propanamide
1-[(6-methoxypyridin-3-yl)methyl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
3-(but-2-yn-1-yl)-5-[1-(1-methylcyclopropanecarbonyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
4-cyclopentanecarbonyl-2-(2-phenylethyl)morpholine
N-cyclopentyl-1-methyl-5-[4-(thiophen-2-yl)butanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(propan-2-yl)-1-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-1H-imidazole
N-{[1-(quinolin-2-ylmethyl)piperidin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
2-methyl-6-[(3R,5S)-5-(pyrrolidine-1-carbonyl)piperidine-3-carbonyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-(2-methoxyacetyl)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-3-carboxamide
5-[4-(1-ethyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]-6-phenyl-2,3-dihydropyridazin-3-one
3-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}(methyl)amino)propan-1-ol
2-(prop-2-en-1-yl)-9-{[2-(propylamino)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
1-{2-[({3-[3-(4-ethylpiperazin-1-yl)-2-hydroxypropoxy]phenyl}methyl)amino]ethyl}piperidin-2-one
(1R,7S)-3-[(4-fluorophenyl)methyl]-6-(thiomorpholine-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
5-[3-(piperidine-1-carbonyl)phenyl]pyrazin-2-amine
2-(cyclohex-1-en-1-yl)-N-[(5-methyl-1,2-oxazol-3-yl)methyl]acetamide