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methyl 9-[(4-fluorophenyl)methoxy]-3-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-cyano-N-[2-(2-ethoxyphenoxy)ethyl]-N-methylbenzamide
4-[(3-hydroxy-4-methoxyphenyl)methyl]-1-(4-methoxyphenyl)piperazin-2-one
2-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)phenyl]-5-methyl-1,3,4-oxadiazole
N-{[1-(2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)piperidin-3-yl]methyl}pyridine-3-carboxamide
3-[(1-benzylpiperidin-4-yl)oxy]-N-(pyridin-3-ylmethyl)benzamide
1,4-dimethyl-9-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-1,4,9-triazaspiro[5.5]undecane
2-[(3-methoxyphenyl)amino]-N-[2-(2-oxoimidazolidin-1-yl)ethyl]butanamide
N-methyl-N-[2-(methylamino)ethyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
methyl 2-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}pyridine-3-carboxylate
5-(2-chloro-4-methoxyphenoxymethyl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1,2-oxazole-3-carboxamide
6-methyl-2-[({[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}amino)methyl]quinolin-4-ol
2-(4-chlorophenyl)-5-[1-(prop-2-en-1-yl)-1H-imidazol-2-yl]pyrimidine
1-cyclopropyl-3-{2-[4-(3,5-dimethylphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)pyrrolidine-2,5-dione
N-(2-{[2-(morpholin-4-yl)ethyl]carbamoyl}phenyl)pyrrolidine-3-carboxamide
4-{2-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]phenyl}morpholine
3-cyclohexyl-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
3-methyl-5-[(2S)-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl]-1,2,4-oxadiazole
1-methyl-N-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-indole-2-carboxamide
N-({7-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)methanesulfonamide
(2,1,3-benzothiadiazol-5-ylmethyl)[1-(diethylamino)propan-2-yl]amine
N-[2-(1H-imidazol-1-yl)ethyl]-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
(1R,5R)-3-methanesulfonyl-6-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-[(4-fluorophenyl)methyl]-2-oxo-1-(pyridin-4-ylmethyl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
3-[(4-ethylpiperazin-1-yl)methyl]-7-methyl-1-propyl-1,2-dihydroquinolin-2-one
N-{[8-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}cyclohexanecarboxamide
6-ethyl-1-methyl-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
8-(3-chloro-4-propoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1-(2,2-dimethylpent-4-en-1-yl)-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
(2S)-2-{[5-(2-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}-3-methylbutanamide
3-(4-fluorophenyl)-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1H-pyrazole-5-carboxamide
N-[(1-hydroxycyclohexyl)methyl]-2-[2-(morpholin-4-ylmethyl)-4-(pyrazin-2-yl)phenoxy]acetamide
2-(1-butyl-1H-pyrazol-4-yl)-8-methyl-4-(morpholine-4-carbonyl)quinoline
5-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
4-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}-1,2-dihydroisoquinolin-1-one
(4aR,7aS)-1-acetyl-4-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1-(propan-2-yl)piperidine-3-carboxamide
N-cyclopentyl-2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
(2E)-1-[3-(4-chlorobenzoyl)piperidin-1-yl]-3-(pyridin-2-yl)prop-2-en-1-one
3-{2-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-oxoethyl}-1-methylimidazolidine-2,4-dione
N-(1,4-dioxan-2-ylmethyl)-N,1-dimethyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-phenyl-N-(pyridin-2-ylmethyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-(2-methoxyethyl)-1-(pyridin-2-yl)-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-{1-[(2-fluorophenyl)methyl]-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperazin-2-yl}ethan-1-ol
4-{4-[3-(propoxymethyl)pyrrolidin-1-yl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-yl}pyridine
N-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
4-[2-oxo-4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]benzonitrile
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-5-(methoxymethyl)-N-methyl-1,3,4-oxadiazole-2-carboxamide
(4aS,8aR)-1-(4-hydroxybutyl)-6-(3,3,3-trifluoropropyl)-decahydro-1,6-naphthyridin-2-one
5-(2,4-difluorophenoxymethyl)-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-1,2-oxazole-3-carboxamide