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2-[1-cyclopentyl-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(propan-2-yl)acetamide
N-(1-{7-[(3,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-2-methoxyacetamide
methyl 4-{[3-(2-ethyl-5-oxopyrrolidin-2-yl)propanamido]methyl}benzoate
2-butoxy-1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
5-methyl-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-2-carboxamide
2-{4-[3-(3,4-difluorophenyl)propanoyl]-2-oxopiperazin-1-yl}benzonitrile
methyl({[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl})({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amine
1-(cyclohexylmethyl)-3-({[(5-fluoro-1H-indol-2-yl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3-dimethoxybenzamide
N-[(3-chlorophenyl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-methyl-4-(4-{[3-(phenylamino)piperidin-1-yl]methyl}phenyl)but-3-yn-2-ol
(3S)-4-(1-benzofuran-3-carbonyl)-3-ethylmorpholine
4-{[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]methyl}-N-methylbenzamide
2-(2-{[methyl({[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})amino]methyl}phenoxy)acetic acid
N-[(3S,4R)-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
ethyl({[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(2-methylprop-2-en-1-yl)amine
({4-ethyl-5-[1-(4-methylpiperazine-1-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
5-chloro-2-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-3-phenyl-1H-indole
{1-[4-(4-{[(4-phenyl-1,3-thiazol-5-yl)methyl]amino}piperidin-1-yl)benzoyl]piperidin-3-yl}methanol
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)benzamide
3-(1H-1,3-benzodiazol-1-yl)-1-[3-(naphthalene-1-carbonyl)piperidin-1-yl]propan-1-one
methyl 4-{[(2-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}ethyl)amino]methyl}benzoate
(1r,4r)-4-({[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)cyclohexan-1-ol
3-({[(2,6-difluorophenyl)methyl]amino}methyl)-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
N'-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-N,N-dimethylbutanediamide
1-cyclopentyl-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-(1-methyl-1H-pyrazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-hydroxy-2-(pyridin-3-yl)-N-{2-[(2S)-pyrrolidin-2-yl]ethyl}pyrimidine-5-carboxamide
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
4,4,4-trifluoro-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}butanamide
6-(2-fluoro-4-methoxyphenyl)-7-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-fluoro-3-(3-propylmorpholine-4-carbonyl)benzene-1-sulfonamide
1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
(5-{[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]methyl}-2-ethoxyphenyl)methanol
N-(2-hydroxyethyl)-N-methyl-1-{1-[(4-phenylphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]pyrimidin-2-amine
2'-amino-4'-(3,4-dihydroxyphenyl)-7',8'-dihydro-5'H-spiro[piperidine-4,6'-quinoline]-3'-carbonitrile
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}pyrrolidin-2-one
2-[1-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazole
(1S,5R)-3-(4-chloro-3-methylbenzoyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2-methoxyphenyl)-4-[1-(1-methylpiperidine-4-carbonyl)piperidin-3-yl]piperazine
N-(3-{4-[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]piperidin-1-yl}phenyl)pyridine-4-carboxamide
N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-2-carboxamide
5-(furan-3-ylmethyl)-3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
ethyl 2-[(2-{[2-(morpholin-4-yl)ethyl]carbamoyl}phenyl)amino]acetate
2-cyclopropyl-4-hydroxy-N-(oxolan-2-ylmethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]pyrimidine-5-carboxamide
naphthalen-1-yl (9aR)-8-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
3-(4-chlorophenyl)-2-[(4,6-dimethylpyrimidin-2-yl)amino]propan-1-ol
1-(3,5-dimethylphenyl)-4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperazin-2-one
(1S,5R)-6-[(2-chloro-4-fluorophenyl)methyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane