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(1S,4S)-5-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
3-[(4aS,7aR)-4-(2-methoxyacetyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]benzonitrile
2-(dimethyl-1H-1,2,4-triazol-1-yl)-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)acetamide
N-{[1-(1H-pyrazole-4-carbonyl)piperidin-3-yl]methyl}-3-(trifluoromethyl)benzamide
(1S,5R)-6-benzyl-3-[(2,3-difluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-chloro-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-5-(trifluoromethyl)benzamide
7-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]acetyl}-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[(3-ethoxy-4-methoxyphenyl)methyl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
N-[2-(2,4-difluorophenyl)-1-{1-[(2E)-3-(2,4-difluorophenyl)prop-2-enoyl]piperidin-4-yl}ethyl]-N-methylpropanamide
3-{2-[(3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
5-(3-fluorophenoxymethyl)-3-(3-phenoxyazetidine-1-carbonyl)-1H-pyrazole
2-[4-(4-fluorophenyl)-2-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy]-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
2-[2-(dimethylamino)ethyl]-8-(5-phenyl-1,2,4-oxadiazol-3-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-(4-chloro-1H-pyrazol-1-yl)-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]propanamide
1-ethyl-8-(1-methoxypropan-2-yl)-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-cyano-N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}benzamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N,3-dimethylthiophene-2-carboxamide
2-methyl-4-(3-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}phenyl)butan-2-ol
2-(dimethylamino)-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-methylpyrimidine-5-carboxamide
4-[(1E)-3-[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]prop-1-en-1-yl]-2-methoxyphenol
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-2,3-dihydro-1-benzofuran-5-carboxamide
(4aS,8aR)-6-(furan-3-ylmethyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-{[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]methyl}benzoic acid
5-[2-(pyrrolidine-1-carbonyl)phenoxy]-1-azabicyclo[3.2.1]octane
4-benzyl-3-ethyl-1-(3-hydroxy-4-methylbenzoyl)-1,4-diazepan-5-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-[(3-chlorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
3-(2-fluorobenzenesulfonyl)-9-methyl-3,9-diazaspiro[5.6]dodecane
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]amine
ethyl 1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-[(propan-2-yl)carbamoyl]pyrrolidine-2-carboxylic acid
2-{4-[3-(4-benzylpiperidin-1-yl)-3-oxopropyl]piperidin-1-yl}acetic acid
5-{1-[(2E)-3-(3,4-difluorophenyl)prop-2-enoyl]piperidin-4-yl}-5-methyl-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
2-[(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenol
1-cyclopropyl-5-{4-[(2-fluorophenyl)methyl]piperidine-1-carbonyl}piperidin-2-one
2-(2-{1-[2-(2,3-dihydro-1H-indol-1-yl)-2-oxoethyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
3-{2-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
4-methyl-6-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}pyrimidin-2-amine
(2S,4S)-1-benzyl-N-methyl-4-{[(3-phenoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
7-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)-3-methyl-3,4-dihydroquinazolin-4-one
9-methoxy-3-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-10-(thiomorpholine-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
2-{[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]amino}-1-phenylethan-1-ol
(1R,5R)-6-(cyclopropylmethyl)-3-(3,5-dimethyl-1-benzofuran-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(pyridin-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-cyclopropyl-4-methoxy-3-{[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]oxy}benzamide
1-(2-methoxyethyl)-4-[4-(thiophen-2-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
4-methyl-2-{2-oxo-2-[2-(pyridin-2-yl)piperidin-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
N-butyl-N-cyclopentyl-1-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
2-{2-[(3,4-dimethylpiperazin-1-yl)methyl]phenoxy}-1-(4-methylpiperidin-1-yl)ethan-1-one
(3R,4R)-1-{[2-(benzylamino)pyrimidin-5-yl]methyl}-4-(hydroxymethyl)piperidin-3-ol
2-amino-6-(1,3-dimethyl-1H-pyrazol-4-yl)-4-[2-(prop-2-en-1-yloxy)phenyl]pyridine-3-carbonitrile