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4-[(2-fluorophenyl)methyl]-3-propyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(3-ethoxy-4-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-[(3-chlorophenyl)methyl]-1-(pyrimidin-2-yl)piperidine-3-carboxylic acid
4-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
5-oxo-1-(pyridin-2-ylmethyl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]pyrrolidine-3-carboxamide
ethyl 4-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperazine-1-carboxylate
4-amino-6-fluoro-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}quinoline-3-carboxamide
3-(1-hydroxyhexan-2-yl)-5-methyl-3,4-dihydroquinazolin-4-one
1-(2-{[(5-chloro-2,4-dimethoxyphenyl)methyl](methyl)amino}ethyl)piperidin-2-one
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-6-phenylpyridazine
1-[(4-methanesulfonylphenyl)methyl]-2-(pyrrolidin-1-ylmethyl)piperidine
1-methyl-1-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}-3-(2,4,6-trimethylpyridin-3-yl)urea
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-3-(1-methylpiperidin-3-yl)propanamide
2-(1-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1,3-benzothiazole
5-cyclopropyl-N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,3,4-oxadiazol-2-amine
3-(4-methoxyphenyl)-N-[1-(pyridin-3-yl)propan-2-yl]-1H-pyrazole-5-carboxamide
(2S,4S)-4-amino-N-methyl-1-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}pyrrolidine-2-carboxamide
2-ethyl-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]pyrimidine-5-carboxamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(piperidin-1-ylmethyl)piperidine
benzyl(methyl)({3-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecane-4-carbonyl]-1,2-oxazol-5-yl}methyl)amine
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(piperidin-1-yl)acetamide
1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)ethan-1-one
5-{1-[(dimethyl-1,3-thiazol-5-yl)methyl]pyrrolidin-2-yl}-N-(1-methyl-1H-1,2,4-triazol-3-yl)thiophene-2-carboxamide
N-(2-{4-[({[5-(methoxymethyl)furan-2-yl]methyl}(methyl)amino)methyl]-5-methyl-1,3-oxazol-2-yl}phenyl)methanesulfonamide
2-(adamantan-1-yl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}acetamide
N-(cyclobutylmethyl)-N-(oxolan-2-ylmethyl)-3-propanamidobenzamide
6-[({2-[(4-chlorophenyl)sulfanyl]ethyl}amino)methyl]-1,4-oxazepan-6-ol
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-3,5-dimethyl-1H-indole-2-carboxamide
2-(3-{[7-(3,4-dihydronaphthalen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenoxy)ethan-1-ol
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-[(5-methylthiophen-2-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
1-(1-phenylpiperidin-4-yl)-1,4-diazepane-6-carboxylic acid
4-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}-1-(furan-2-carbonyl)piperidine
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
5-(2H-1,3-benzodioxol-5-yl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1,2,4-triazin-3-amine
1-(furan-2-ylmethyl)-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
3-[2-(methylsulfanyl)benzoyl]-1-(oxan-4-yl)piperidine
methyl 5-[(cyclohex-3-en-1-ylmethyl)amino]-1-(2-methoxyethyl)-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(3-hydroxyphenyl)-N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-5-oxopyrrolidine-3-carboxamide
3-(3-methyl-1H-pyrazol-1-yl)-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
N,N-dimethyl-7-(4-methyl-1H-imidazole-5-carbonyl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-methyl-N-[(1S,3S)-3-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}cyclopentyl]-1H-pyrrole-2-carboxamide
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(propan-2-yl)piperidine
2-{[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1-methyl-1H-1,3-benzodiazole
3-(3,4-dimethoxybenzoyl)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine
7-(morpholin-4-ylmethyl)-4-(naphthalen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
{4-[(dimethylamino)methyl]-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}methanol
3-(2,3-dihydro-1H-inden-2-yl)-5-{1-[(2E)-3-(1H-imidazol-4-yl)prop-2-enoyl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-N,N-dimethylpyrimidin-4-amine
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-{imidazo[1,2-a]pyrimidine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane