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1-{2,7-diazaspiro[4.5]decan-2-yl}-2-[(2-methylphenyl)amino]ethan-1-one
N-methyl-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-N-[2-(1H-pyrazol-4-yl)ethyl]pyridin-2-amine
6-(2-aminoethyl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-4-amine
1-({[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)propan-2-ol
2-cyclopropyl-9-[4-(trifluoromethyl)pyridin-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(2S,4R,6R)-2-(diphenylmethyl)-6-(propan-2-yl)oxan-4-yl]acetamide
[4-(1,3-benzoxazol-2-yl)-1,4-oxazepan-6-yl]methanol
1-(1H-imidazol-2-ylmethyl)-5-(pentan-2-yl)-4-phenyl-1H-imidazole
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
[(2S,4R,5R)-5-(2-fluorophenyl)-4-({[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]amino}methyl)-1-methylpyrrolidin-2-yl]methanol
2-methyl-3-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1,2,3,4-tetrahydroisoquinoline
9-(4-ethyl-5-methylpyrimidin-2-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-2-(1,3-thiazol-4-yl)acetamide
2-{4-[(5-chloro-2,3-dimethoxyphenyl)methyl]piperazin-1-yl}-N,N-dimethylacetamide
4-(2-methylphenoxy)-1-(oxane-4-carbonyl)piperidine-4-carboxylic acid
1-[7,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carbonyl]-N,N-dimethylpiperidin-3-amine
N,N-diethyl-1-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carboxamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
N6-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N5,N5-dimethyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-methyl-8-[4-(2-methylpropyl)benzoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-ethyl-3-oxo-N-[(1R)-1-phenylpropyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
10-(3-hydroxypiperidine-1-carbonyl)-9-methoxy-3-[(4-methoxy-2,5-dimethylphenyl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
3-(oxolan-3-yl)-1-(2,3,5-trifluorophenyl)urea
2-[4-(methylsulfanyl)phenyl]-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]acetic acid
4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidine
(4aR,8aS)-6-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-1-{[4-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
(3aR,6aR)-2-acetyl-5-(2,1,3-benzoxadiazol-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-({[2-(3-fluorophenyl)ethyl]amino}methyl)-4-phenylphenol
2-methanesulfonamido-N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}acetamide
N-ethyl-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridin-2-amine
N-[(2R,3R)-2-methoxy-1'-[2-(piperidin-1-yl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
2-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-2-yl}pyridine
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}[2-(methylsulfanyl)ethyl]amine
1-(furan-2-yl)-2-[(3S,4S)-3-hydroxy-4-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}pyrrolidin-1-yl]ethane-1,2-dione
5-(4-acetylphenoxymethyl)-N-methyl-N-[2-(morpholin-4-yl)ethyl]-1,2-oxazole-3-carboxamide
(2S,4R)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-[(4-methoxyphenyl)sulfanyl]-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]acetamide
3-{2-oxo-2-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]ethyl}-1,3-oxazolidin-2-one
2-{1-[(6-ethoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidin-2-yl}acetamide
N-[(2R,3R)-1'-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
(4aS,8aR)-6-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
3-methyl-3-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-1-[3-(pyridin-2-yl)phenyl]urea
(4aR,7aS)-1-(cyclopropylmethyl)-4-(1H-imidazol-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-(3-chloro-4-methylbenzoyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
2-(2H-1,3-benzodioxol-5-yloxy)-1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-cyclopentyl-4-[2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]piperazine
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-{[4-(4-fluorophenoxy)piperidin-1-yl]methyl}pyridin-2-amine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide