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2-[4-(propan-2-yl)morpholin-2-yl]-N-[(4-sulfamoylphenyl)methyl]acetamide
(3R,5S)-N3-(4-fluorophenyl)-1-(2-methylpropyl)-N5-(oxolan-2-ylmethyl)piperidine-3,5-dicarboxamide
2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(pyridin-2-ylmethyl)acetamide
2-(4-chlorophenyl)-4-[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]morpholine
7-[(2-fluorophenyl)methyl]-2-(1,2,3-thiadiazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(2-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-4-(pyrimidin-5-yl)phenoxy)acetic acid
1-[4-(oxan-4-yl)piperazin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
1-(2-cyclopropylacetyl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(3,5-difluorophenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(3,4-dimethoxyphenyl)ethyl]-3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanamide
5-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-N-ethylpyrimidin-2-amine
1-(piperidin-1-yl)-N-[2-(pyridin-3-yl)ethyl]cyclohexane-1-carboxamide
N,2,6,8-tetramethyl-N-[2-(2-oxopiperidin-1-yl)ethyl]quinoline-4-carboxamide
methyl 2-{8-benzyl-1-[2-(4-methoxyphenyl)ethyl]-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-1-(4-ethylpiperazin-1-yl)propan-1-one
N-cyclopropyl-N-({3-[(2-fluorophenyl)methoxy]phenyl}methyl)-4-methylbenzamide
7-[2-(5-methoxy-1H-indol-3-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
(2S,4R)-N-[2-(4-fluorophenyl)ethyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
N-[(2R,3R)-1'-(1-benzofuran-2-ylmethyl)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
ethyl 4-{1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidin-3-yl}piperazine-1-carboxylate
methyl (2S,4S)-1-(quinolin-4-ylmethyl)-4-(thiophene-2-amido)pyrrolidine-2-carboxylate
6-(4-cyclopentylpiperazine-1-carbonyl)-2-(3-methoxyphenyl)-1,3-benzoxazole
1-methyl-2-[1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-3-yl]-1H-1,3-benzodiazole
(2S)-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-acetamidopropanamide
N-(2-fluorophenyl)-3-[1-(6-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)piperidin-3-yl]propanamide
{2-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}urea
2-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]-N-(1-methyl-1H-pyrazol-3-yl)acetamide
4-[4-(1H-imidazol-1-yl)benzoyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
1-(3,5,7-trimethyl-1H-indole-2-carbonyl)piperidine-3-carboxylic acid
N-[1-({[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]furan-2-carboxamide
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
7-methoxy-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
methyl (2S)-1-[(4-benzyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]pyrrolidine-2-carboxylate
3-(3-chlorophenyl)-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-3-phenylpropanamide
7-(cyclopropylmethyl)-2-{[3-(methylsulfanyl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
3-(3-methoxypropyl)-1-(6-oxo-1,6-dihydropyridazine-3-carbonyl)piperidine-3-carboxylic acid
2-[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole
(3R,4R)-1-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-3,4-dimethylpyrrolidin-3-ol
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
N,N,2-trimethyl-7-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-[2-(dimethylamino)ethyl]-5-[1-(3-methylbenzoyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-[(2-chlorophenyl)methyl]-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-1,4-diazepan-5-one
4-(2,7,8-trimethylquinoline-4-carbonyl)-1,4-oxazepan-6-ol
N'-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)pentanediamide
1-(4-cyclopentyl-1,4-diazepan-1-yl)-2-(2,5-dimethoxyphenyl)ethan-1-one
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrimidine-4-carboxamide
[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl){[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl}amine
7-[(2,3-difluorophenyl)methyl]-2-(furan-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
methyl 9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxylate