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2-({[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)amino)-1-phenylethan-1-ol
3-(3-chlorophenyl)-N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-3-phenylpropanamide
1-{4-[(4aR,8aS)-6-(4-phenylbutanoyl)-decahydro-1,6-naphthyridine-1-carbonyl]phenyl}pyrrolidin-2-one
methyl({[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
N-[2-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]pyridine-3-carboxamide
N-{1-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-4-yl]-2-phenylethyl}-N-methylthiophene-3-carboxamide
N-(furan-2-ylmethyl)-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
2-(cyclopentylmethyl)-1-(2-methoxyethyl)-6-methyl-4-oxo-N-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
methyl (2S,4S)-4-(2-benzyl-1,3-thiazole-4-amido)-1-methylpyrrolidine-2-carboxylate
1-[(4-methyl-1H-imidazol-5-yl)methyl]-8-(quinolin-6-yl)-1,8-diazaspiro[4.5]decane
methyl 3-(3,4-difluorobenzoyl)-9-[2-(1-methylpyrrolidin-2-yl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-{[8-(2-phenylethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
(4aS,8aR)-6-methanesulfonyl-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
N-methyl-5-[3-(1-methylpiperidin-3-yl)propanoyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,6-difluorobenzamide
4,6-dimethyl-5-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-1-carbonyl)-2H-pyran-2-one
2-(4,5-dichloro-2-methyl-1H-imidazol-1-yl)-N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
2-[3-(1H-imidazol-1-yl)propyl]-3-oxo-N-(propan-2-yl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-methyl-N-[1-(2-phenylacetyl)azepan-3-yl]-1H-imidazole-4-sulfonamide
3-[3-phenyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydroquinoxalin-2-one
5-{[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}-2-hydroxybenzoic acid
4-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-6-(pyrrolidin-1-yl)pyrimidine
(4aS,7aR)-1-[3-(1H-pyrazol-1-yl)propanoyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(benzenesulfonyl)-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
3-[1-(2-phenylethyl)piperidin-4-yl]propanoic acid
N,2-diethyl-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]pyrimidine-5-carboxamide
8-[(3-chloro-4-hydroxyphenyl)methyl]-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-[methyl(1-methylpiperidin-4-yl)amino]ethan-1-one
[2-(1,3-benzothiazol-2-yloxy)hex-5-en-1-yl]dimethylamine
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-1-ethyl-3-methylpiperidine-3-carboxamide
N-[3-(dimethylcarbamoyl)-5-({[(4-ethylphenyl)methyl]amino}methyl)phenyl]pyridine-2-carboxamide
2,5-dimethoxy-N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]benzamide
1'-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-(2-{[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
4-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-2-ethyl-1-(propan-2-yl)piperazine
N-({1-[(3-cyanophenyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)-2-methylbenzamide
1-{2-[(4-fluorophenyl)methyl]morpholin-4-yl}-2-(pyridin-4-ylsulfanyl)ethan-1-one
4-{[(furan-2-ylmethyl)(prop-2-en-1-yl)amino]methyl}-2,6-dimethylphenyl acetate
3-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]amino}pyrazine-2-carbonitrile
(3S)-2-(2-aminopyridine-4-carbonyl)-N-tert-butyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-(4-cyanonaphthalen-1-yl)-3-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]urea
5-benzyl-4-[1-(2-fluorobenzoyl)piperidin-3-yl]-2-methylpyrimidine
5-methyl-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(propan-2-yloxy)phenyl]methyl}thiophene-2-carboxamide
[(1-ethylpiperidin-3-yl)methyl]({[4-(1H-imidazol-1-yl)phenyl]methyl})methylamine
2-methoxyethyl N-{[(2S,4S)-4-fluoro-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}pyrrolidin-2-yl]methyl}carbamate
2-[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]pyridine-4-carboxamide
2-phenoxy-N-{[7-(quinolin-4-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}acetamide
8-[1-(morpholin-4-yl)cyclohexanecarbonyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(2-{[4-(3-hydroxyphenyl)piperidin-1-yl]methyl}phenyl)-6-methyl-3,4-dihydropyrimidin-4-one
1-{5-[3-(pyrazin-2-yl)-1H-pyrazol-1-yl]-1H-1,3-benzodiazol-2-yl}ethan-1-ol