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3-(azetidine-1-carbonyl)-N-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]benzene-1-sulfonamide
4-({[(1S,2S)-2-hydroxycyclohexyl]carbamoyl}amino)-N-(2-phenylethyl)benzamide
N-[(5-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
1-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-2,1-benzoxazole-3-carboxamide
N-(3-{2-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-1H-imidazol-1-yl}phenyl)methanesulfonamide
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(6-methylpyridin-2-yl)piperidine-4-carboxylic acid
N-{2-[2-(2-cyclohexylpyrimidin-5-yl)-1H-imidazol-1-yl]ethyl}-2-methylpropanamide
6-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]pyridine-3-carboxylic acid
9-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-[2-(5-methyl-1H-pyrazol-1-yl)ethyl]-3-(2-methylpropyl)-1-phenyl-1H-1,2,4-triazole
9-(2-fluoro-4-methylbenzenesulfonyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
1-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
5-({5-[(2E)-but-2-en-1-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
2-{[2-(2-carboxyethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]methyl}-1,3-oxazole-4-carboxylic acid
6-[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
1-(6-methylpyridine-2-carbonyl)spiro[azepane-4,2'-chromene]
N-[2-hydroxy-2-(pyridin-4-yl)ethyl]-3-(3-hydroxy-3-methylbutyl)benzamide
(6R)-6-[4-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1,3-diazinane-2,4-dione
1-(3-chlorophenyl)-4-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]piperazine
5-[3-(1,2-oxazinan-2-yl)propanoyl]-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
3,5-difluoro-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-2,6-dimethylquinoline-4-carboxamide
(2S)-2-({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}amino)propanamide
1-(4-fluoro-3-methoxyphenyl)-3-[(1-methyl-4-phenylpiperidin-4-yl)methyl]urea
N-cyclopropyl-5-[(4-hydroxypiperidin-1-yl)methyl]-N-(2-methylpropyl)-1,2-oxazole-3-carboxamide
3-(2-chlorophenyl)-1-{3-[4-(3,4-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
methyl 2-[8-(cyclohex-3-en-1-ylmethyl)-1-(2-methoxyethyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
1-(furan-3-carbonyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
7-(1,3-benzothiazol-2-yl)-4-cyclopentanecarbonyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[4-(pyridin-4-yl)piperazine-1-carbonyl]morpholine
2-(2,3-difluorophenyl)-N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}acetamide
1-[3-(2-{[(cyclopropylmethyl)(methyl)amino]methyl}-4-methoxyphenoxy)-2-hydroxypropyl]piperidin-4-ol
(2R,3R)-2-hydroxy-3-(1H-imidazol-1-yl)-N-phenyl-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-carboxamide
8-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-8-azaspiro[4.5]decane-7,9-dione
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-4-(4-methoxyphenyl)butane-1,4-dione
6-{4-[(8-methylquinolin-5-yl)methyl]piperazin-1-yl}pyridine-2-carbonitrile
3-methoxy-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]benzamide
1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-3-(furan-2-yl)propan-1-one
2,5-difluoro-N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
3-[1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-2-yl]propan-1-ol
2-methoxy-1-[9-(oxolan-3-ylmethoxy)-7-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
(1,3-benzoxazol-2-ylmethyl)({[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
N-methyl-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]acetamide
3-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-2H-chromen-2-one
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
1-(2-{[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]amino}pyrimidin-4-yl)piperidin-3-ol