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N-[1-(3-methylphenyl)piperidin-4-yl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
1-({2-[2-hydroxy-3-(thiomorpholin-4-yl)propoxy]phenyl}methyl)piperidine-4-carbonitrile
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidine-4-carboxylic acid
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-[(2E)-3-phenylprop-2-enoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
1-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
N-{[5-chloro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methyl-1H-indol-3-yl)acetamide
4-(1-butyl-1H-imidazol-2-yl)-1-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}piperidine
2-{[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]methyl}-8-fluoro-1,4-dihydroquinolin-4-one
3-(5-fluoro-2-methoxybenzoyl)-N-(4-fluorophenyl)piperidine-1-carboxamide
9-(1H-1,2,3-benzotriazole-5-carbonyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-cyclopropyl-N-{2-[4-(dimethylamino)phenyl]ethyl}pyrimidine-5-carboxamide
(4aS,8aS)-2-{[2-(trifluoromethoxy)phenyl]methyl}-decahydroisoquinolin-4a-ol
1-(4-phenylpiperazine-1-carbonyl)-6-(3-phenylpropyl)-6-azaspiro[2.5]octane
N-({8-[(2-methylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-4-oxo-4H-chromene-2-carboxamide
2-{[4-(4-methoxyphenyl)piperazin-1-yl]methyl}-6-methylquinazolin-4-amine
5-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-5-(pyridin-2-yl)imidazolidine-2,4-dione
[(3R,4R)-1-(5-methyl-1,3-oxazole-4-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-3-methylthiophene-2-carboxamide
9-[(4-chloro-3-fluorophenyl)methyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-2-(furan-2-yl)pyrimidine
1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-(1-methyl-1H-indol-3-yl)ethan-1-one
N-({1-[(5-ethylpyridin-2-yl)methyl]piperidin-3-yl}methyl)-1H-pyrrole-2-carboxamide
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-6-fluoro-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-(3-aminoazepan-1-yl)-3-(2,3-dihydro-1H-indol-1-yl)propan-1-one
1-(1-benzylpiperidin-4-yl)-N-ethyl-N-methylpiperidine-3-carboxamide
4-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-4-oxobutane-1-sulfonamide
2-[3-(2-methoxyethyl)-5-(1-methyl-1H-pyrazol-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
4-{4-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]piperazin-1-yl}-5,6-dimethylpyrimidine
5-[1-(3,5-difluorobenzoyl)piperidin-4-yl]-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
2-(2-fluorophenyl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-{[4-(cycloheptyloxy)-3-methoxyphenyl]methyl}-N-(pyridin-2-ylmethyl)-2-(thiophen-3-yl)acetamide
methyl 3-(2,3-dimethylbenzoyl)-9-[2-(morpholin-4-yl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-6-(trifluoromethyl)pyridin-2-ol
1-{2-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-oxoethyl}pyrrolidin-2-one
N5-cyclopentyl-N6-(prop-2-en-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
5-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
1-[5-amino-2-ethyl-1-(3-methoxypropyl)-1H-1,3-benzodiazole-7-carbonyl]-4-(4-chlorophenyl)piperidin-4-ol
(2S,4S)-4-amino-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}pyrrolidine-2-carboxylic acid
N-methyl-1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
N4-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-(2-methoxy-5-methylphenyl)-3-{[1-(oxan-4-yl)pyrrolidin-3-yl]methyl}urea
6-oxo-N-[4-(oxolan-2-yl)butyl]-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
3-(3-methylbutyl)-8-{spiro[2.4]heptane-1-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[3-(2-methoxybenzoyl)piperidin-1-yl]propanoic acid
N-cyclopentyl-3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(pyridin-4-ylmethyl)piperidin-3-yl]propanamide
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]quinoxaline
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-4-(methoxymethyl)-N-methylpiperidine-1-sulfonamide