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N-ethyl-3-(methylsulfanyl)-N-{[3-(prop-2-en-1-yloxy)phenyl]methyl}propanamide
2-(morpholin-2-yl)-N-[(3-phenylphenyl)methyl]acetamide
2-methoxy-4-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
5-acetamido-1-ethyl-2-(2-fluorophenyl)-N-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
1-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(3-methylphenoxymethyl)piperidine
N-benzyl-2-[3-(2-methoxyphenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-(2-phenylethyl)acetamide
6-[(5-methyl-1,2,4-oxadiazol-3-yl)methoxy]-4-[(1-methyl-1H-indol-3-yl)methyl]-1-(propan-2-yl)-1,4-diazepan-2-one
(2S)-2-{[2-(dimethylamino)-6-methylpyrimidin-4-yl]amino}-3-phenylpropanamide
5-{3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl}pyridine-2,4-diol
5-[1-(5-acetylthiophene-3-carbonyl)piperidin-4-yl]-5-ethyl-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
ethyl 4-(2-phenoxyethyl)-1-(pyridin-4-ylmethyl)piperidine-4-carboxylate
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
2-(2-methyl-1H-imidazol-1-yl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-(dimethyl-1,2-oxazol-4-yl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}propan-1-one
(4aS,8aR)-1-(2-aminoethyl)-6-[(5-chlorothiophen-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
1-ethyl-5-{[(1-ethylcyclobutyl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-(3-hydroxyphenyl)-1-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]ethan-1-one
N-(1-hydroxy-3-methylbutan-2-yl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
7-(2,6-dimethoxyphenyl)-9-methoxy-4-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(1-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
(4aS,7aR)-N-ethyl-4-[(4-methyl-1H-imidazol-5-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
4-({1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl}methyl)morpholine
N-methyl-3-(pyridin-2-yl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]propanamide
5,6,7-trimethoxy-4-(1-methyl-1H-1,2,3-benzotriazol-5-yl)-1,2,3,4-tetrahydroquinolin-2-one
N-methyl-4-{[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}benzene-1-sulfonamide
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-(2,2-dimethyloxan-4-yl)pyrrolidin-2-one
7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-4-(quinolin-5-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2,1,3-benzoxadiazol-5-ylmethyl)[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]methylamine
3-{2-[3-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-1-(2-methoxyethyl)-3-(2-methoxyphenyl)pyrrolidine-2,5-dione
1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(N-methylmethanesulfonamido)ethyl]benzamide
4-ethyl-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,2,3-thiadiazole-5-carboxamide
2-[1-benzyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
1-(cyclopropylmethyl)-5-(2-methoxybenzoyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1'-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(diethylcarbamoyl)methyl]-N-(3,3-diphenylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-cyclopropyl-5-[3-(morpholin-4-ylmethyl)phenyl]thiophene-2-carboxamide
(1S,9R)-11-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
5-(5-chloro-2-methoxyphenyl)-2,4-dimethoxypyrimidine
1-(1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-1H-pyrazole-4-carbonyl)-N,N-diethylpyrrolidin-3-amine
methyl (2S)-1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxylate
3-[4-(adamantan-1-yl)piperazine-1-carbonyl]-2-ethyl-1-[(4-methoxyphenyl)methyl]-6-methyl-1,4-dihydropyridin-4-one
2-{2-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-2-oxoethyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one
3-[3-(1,2-oxazol-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{1-[(2Z)-3-(3-fluorophenyl)prop-2-enoyl]piperidin-4-yl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N,N-dimethyl-6-{[1-(morpholin-4-yl)hex-5-en-2-yl]oxy}pyrazin-2-amine
N-(2-hydroxyethyl)-2-[2-(1-methyl-1H-imidazol-4-yl)ethyl]-1-oxo-2,3-dihydro-1H-isoindole-4-carboxamide
1-ethyl-N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)-1H-pyrazole-4-sulfonamide