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1-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperidin-3-ol
2-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonane-7-carbonyl]thiophene-3-sulfonamide
(2S,4R)-4-amino-1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-N-methylpyrrolidine-2-carboxamide
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(pyridin-3-yl)propyl]acetamide
(5S,9aS,9bS)-2-cyclopentyl-5-(3-methylthiophen-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-(2H-1,3-benzodioxole-5-carbonyl)-1-benzyl-6-methoxy-1,4-diazepan-2-one
3-[4-(2,5-difluorophenyl)-1H-pyrazol-5-yl]-1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidine
[1-(oxan-4-yl)-3-(2-phenylethyl)piperidin-3-yl]methanol
methyl 3-{4-[2-(2-fluorophenyl)acetyl]-2-oxo-6-(pyridin-4-ylmethoxy)-1,4-diazepan-1-yl}propanoate
2-cyclohexyl-5-{1-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-1H-imidazol-2-yl}pyrimidine
2-(2-methoxyethyl)-6-[(2S)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl]-1,3-benzoxazole
[(3R,4R)-1-[(4-fluoro-3-methoxyphenyl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-{[3-(2-chlorophenyl)-1,2-oxazol-5-yl]methyl}-5-cyclopropyl-1,3,4-oxadiazol-2-amine
6-ethyl-N-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
9-[(3-ethoxy-4-methoxyphenyl)methyl]-6-oxa-9-azaspiro[4.5]decane
1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
6-[2-fluoro-6-(propan-2-yloxy)phenyl]pyrimidin-4-amine
2-(1H-imidazol-4-yl)-1-(4-methoxy-2-methylphenyl)-1H-imidazole
2-methoxy-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)acetamide
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-8-(1-propylpiperidin-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-cyclopentyl-N-{1-[(3-methylphenyl)methyl]cyclopropyl}-5-oxopyrrolidine-3-carboxamide
4-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-2-[(3-methoxyphenyl)methyl]morpholine
2-methoxy-1-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
3-{3-[(5-cyano-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl)methyl]-1H-indol-1-yl}propanamide
{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-(4-fluorophenoxy)acetamide
1-(2-cyclohexylethyl)-3-hydroxy-3-{[(pyridin-3-ylmethyl)amino]methyl}piperidin-2-one
N-ethyl-2-(4-fluorophenoxymethyl)-4-hydroxy-N-[(2-methylphenyl)methyl]pyrimidine-5-carboxamide
4-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-4H-1,2,4-triazole
8-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-1-[(2-fluorophenyl)methoxy]-1,8-diazaspiro[4.5]decan-2-one
N-[(3,4-difluorophenyl)methyl]-2-(ethylamino)-4-methyl-1,3-thiazole-5-carboxamide
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-cyclopentylethan-1-one
2-[4-(5-amino-4-chloro-1H-pyrazole-3-carbonyl)-1,4-diazepan-1-yl]-N,N-dimethylacetamide
2-(3,4-dichlorophenyl)-4-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]morpholine
3-(1-{2-[(propan-2-yl)amino]pyrimidine-5-carbonyl}piperidin-3-yl)benzoic acid
2-{4-[3-(1H-indol-3-yl)propanoyl]-2-oxopiperazin-1-yl}benzonitrile
3-{[(4-hydroxyquinolin-2-yl)methyl](methyl)amino}-1λ6-thiolane-1,1-dione
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]propanamide
5-methyl-5-{1-[2-(3-methylphenyl)acetyl]piperidin-4-yl}-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
1-{1-[2-(4-methylphenoxy)acetyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
2-(4-{3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperazin-1-yl)-1,3-benzoxazole
5-(4-phenylazepane-1-carbonyl)-2-(pyridin-3-yl)pyrimidin-4-ol
(benzylsulfamoyl)[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amine
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
1-[3-(5-butyl-4-phenyl-1H-imidazol-1-yl)propyl]piperidine-3-carboxamide
1-(ethanesulfonyl)-4-{4-[(3-propylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}piperidine
1-{[2-(difluoromethoxy)phenyl]methyl}-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
7-(3-hydroxypyridine-2-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}propanamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[2-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]propanamide