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2-(ethoxymethyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-[(3S,4R)-3-cyclopropyl-4-[4-(1H-1,2,4-triazol-1-yl)butanamido]pyrrolidin-1-yl]acetic acid
2-(1-butyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-methyl-N-(oxan-4-yl)acetamide
2-(3-hydroxypropyl)-9-(6-methyl-4-oxo-4H-pyran-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{[ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
2-methyl-N-({5-methyl-2-[2-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)propanamide
1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]-N-(2-phenylethyl)piperidine-4-carboxamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-1-(methoxymethyl)cyclobutane-1-carboxamide
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
methyl (2S,4R)-1-[(2-chloro-6-fluorophenyl)methyl]-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
4-(3,4-diethoxyphenyl)-2-(4-methanesulfonylphenyl)-1H-imidazole
(3S,4R)-1-[(2-chloro-4-fluorophenyl)methyl]-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(4-hydroxyphenyl)propan-1-one
N-[(1-hydroxycyclohexyl)methyl]-2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
2-{[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]methyl}benzoic acid
2,4-dimethoxy-N-{[4-methoxy-3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)benzamide
N-[(3-chlorophenyl)methyl]-3-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}propanamide
[(2-fluoro-5-methoxyphenyl)methyl][(1-methylpiperidin-4-yl)methyl](2-phenylethyl)amine
5-({[(3-{2-[4-(3-methoxybenzoyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
(2S,4S)-4-amino-1-[1-(2,3-dimethylphenyl)piperidin-4-yl]-N-ethylpyrrolidine-2-carboxamide
(3R,4S)-4-[ethyl({[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl})amino]oxolan-3-ol
methyl 7-oxo-3-[2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetyl]-9-(propan-2-yloxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
methyl (2S,4R)-4-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-amido]-1-methylpyrrolidine-2-carboxylate
4,4,4-trifluoro-1-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}butan-1-one
(3S,4S)-4-cyclopropyl-1-{5-[(diethylamino)methyl]-2-methylfuran-3-carbonyl}pyrrolidine-3-carboxylic acid
2-{3-[2-(2-ethylpyrimidin-5-yl)-1H-imidazol-1-yl]phenyl}acetic acid
5-(6-methoxypyridin-3-yl)-3-methylpyridin-2-amine
3,4,7-trimethyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-indole-2-carboxamide
N-methyl-5-(phenoxymethyl)-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-3-carboxamide
methyl 1-[(3R,5S)-5-[(diphenylmethyl)carbamoyl]-1-(furan-2-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-cyclohexyl-N-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]-1H-pyrazole-4-carboxamide
6-ethyl-N-[2-(1H-imidazol-4-yl)ethyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
1-[(2-fluorophenyl)methyl]-6-oxo-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]piperidine-3-carboxamide
N3-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}-N1-(pyridin-3-yl)propane-1,3-diamine
6-({[(1-benzyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)-1,4-oxazepan-6-ol
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-8-[(5-methylthiophen-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(2-methyl-2H-1,2,3-benzotriazol-4-yl)-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)urea
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
2-[4-(2,2-dimethylpropyl)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl]ethan-1-ol
2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}ethan-1-one
N-[(1-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)methyl]naphthalene-1-carboxamide
1-(1-cyclobutanecarbonylpiperidine-4-carbonyl)-2-(1,3-thiazol-2-yl)piperidine
ethyl 4-(2-methoxyethyl)-1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidine-4-carboxylate
(2,1,3-benzoxadiazol-5-ylmethyl)({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
N-cyclopropyl-5-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methylpropyl)acetamide
2-(4-fluorophenyl)-N-(2-{7-[(2-hydroxy-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
(1R,2S)-2-[4-(3-chlorophenyl)-3-oxopiperazine-1-carbonyl]-N-methylcyclohexane-1-carboxamide
1-(2,3-dihydroxypropyl)-N-[3-(furan-2-yl)phenyl]piperidine-4-carboxamide