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N-{1-[1-(furan-3-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N,1-dimethyl-1H-pyrazole-3-carboxamide
5-[(2-fluoro-5-methoxyphenyl)methyl]-5-(3-{4-[hydroxy(phenyl)methyl]piperidin-1-yl}-3-oxopropyl)pyrrolidin-2-one
N-({7-[2-(2-chlorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-sulfonamide
(2S,4R)-N-[(1S)-1-cyclohexylethyl]-4-(3-methoxybenzamido)pyrrolidine-2-carboxamide
5-(4-fluorophenyl)-2-methyl-4-[1-(1-methylcyclohexanecarbonyl)piperidin-3-yl]pyrimidine
(4aR,7aS)-1-ethyl-4-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-propyl-N-{1-[2-(trifluoromethyl)phenyl]ethyl}-1H-pyrazole-5-carboxamide
2-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-pyrrole
(3S,9aR)-2-methyl-3-(2-methylpropyl)-8-(quinolin-5-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(2-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}ethyl)pyridine
1-[5-(methoxymethyl)furan-2-carbonyl]-4-(pyridin-4-yl)piperazine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-(3-hydroxypropyl)-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
6-methyl-4-[3-(oxolan-3-yl)-1-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
N-{[2-(benzyloxy)phenyl]methyl}-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
N-ethyl-1-methyl-N-[2-(4-methylbenzenesulfonyl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
(4aS,7aR)-1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
1-cyclohexyl-N-(furan-2-ylmethyl)-N-(2-hydroxyethyl)piperidine-3-carboxamide
6-[(2E)-3-(2,4-difluorophenyl)prop-2-enoyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
4-{4-[(3-ethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-methylpiperidin-4-ol
N-[2-(dimethylamino)ethyl]-1-{1-[3-(4-methylphenyl)propanoyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
4-[(4-fluorophenyl)methyl]-1-(1H-imidazol-4-ylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
2-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(2,5-difluorophenyl)methyl]acetamide
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
4-oxo-4-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}butanamide
3-{2-[1-ethyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-3,4-dihydroquinazolin-4-one
3-(2,3-dimethylquinoxaline-6-carbonyl)-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
methyl 2-chloro-5-({methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl]carbamoyl}amino)benzoate
2-chloro-6-methoxy-4-({[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amino}methyl)phenol
2-(6-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]acetamide
N-({6-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]pyridin-3-yl}methyl)acetamide
3-(6-methoxynaphthalene-2-carbonyl)-1-[3-(methylsulfanyl)propyl]piperidine
3-(1,3-dihydro-2-benzofuran-5-yl)-1-[4-(furan-2-yl)butan-2-yl]urea
4-(4-hydroxyquinolin-2-yl)-3-methyl-2-propyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-[2-(2,2-diphenylethyl)morpholin-4-yl]-2-methoxyethan-1-one
1-ethyl-6-oxo-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]piperidine-3-carboxamide
4-[3-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}oxy)benzoyl]morpholine
4-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-1λ6-thiane-1,1-dione
1-ethyl-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
5-cyclobutanecarbonyl-1'-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
5-{[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-1,3,4-thiadiazol-2-amine
[2-({4-[(2,3-dimethyl-1H-indol-7-yl)methyl]piperazin-1-yl}methyl)phenyl]methanol
3-(4-methylpiperazine-1-carbonyl)-5-(4-methylpiperidin-1-yl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole
N-methyl-N-(1-methylpyrrolidin-3-yl)-5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
(3S,4R)-1-(2,3-dihydro-1-benzofuran-5-carbonyl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
2-(2,3-difluorophenoxymethyl)-N-[(2R)-1-hydroxybutan-2-yl]-1,3-oxazole-4-carboxamide
2-(2-{1-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-2-yl}ethyl)pyridine
2-ethyl-4-methyl-6-(3,4,5-trimethoxyphenyl)pyrimidine