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1-[4-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)phenyl]ethan-1-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-[3-(3-chlorophenyl)phenyl]-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
1-{2-[3-methyl-4-({[(2-methylphenyl)methyl]amino}methyl)-1H-pyrazol-1-yl]ethyl}piperidin-4-ol
8-[(3-fluoro-2,4-dimethylphenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(5-fluoro-1-methyl-1H-indol-3-yl)methyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
2-{6-chloro-3-[(3-methoxypiperidin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carbonyl}-1,2,3,4-tetrahydroisoquinoline
N,4-dimethyl-2-(propan-2-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]-1,3-thiazole-5-carboxamide
1-[benzyl(methyl)amino]-3-[4-({[(5-ethylpyridin-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
2-amino-1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2-methylpropan-1-one
N-[2-(3-fluorophenyl)ethyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-3-carboxamide
8-acetyl-2-[(3,4-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
3-(4-chlorophenyl)-N-methyl-N-(oxan-4-yl)-3-phenylpropanamide
{3-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-oxopropyl}urea
2-(1-{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-2-yl)ethan-1-ol
2,2-dimethyl-N-{1-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
methyl (2S)-1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxylate
3-(dimethyl-1H-1,2,4-triazol-1-yl)-1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-methylpropan-1-one
N3-[2-(4-fluorobenzenesulfonyl)ethyl]piperidine-1,3-dicarboxamide
(2R,3R,6R)-5-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[5-methoxy-2-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(3-phenylpropyl)propanamide
1-(pyrimidin-2-yl)-4-{5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}-1,4-diazepane
N-({1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]piperidin-3-yl}methyl)-1H-indazole-3-carboxamide
N-[3-(4-{[(2,3-dimethoxyphenyl)formamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-2-methylfuran-3-carboxamide
3-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]benzonitrile
N-[2-(2,4-dimethoxyphenyl)ethyl]-3-(5-phenyl-1,3,4-oxadiazol-2-yl)propanamide
2-{[7-(2-methyl-1,3-thiazole-4-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethan-1-ol
N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}imidazo[1,2-a]pyrimidine-2-carboxamide
N,8-dimethyl-3-({methyl[(1-methylpiperidin-2-yl)methyl]amino}methyl)-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
N-[2-(4-methoxyphenyl)ethyl]-2-methyl-N-[(1-methylpiperidin-4-yl)methyl]-1,3-thiazole-4-carboxamide
4-(1-tert-butyl-1H-pyrrole-3-carbonyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
5-[({4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}formamido)methyl]thiophene-2-carboxylic acid
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[2-(3-methoxyphenyl)piperidin-1-yl]ethan-1-one
methyl (2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-{[2-(pyridin-2-yl)ethyl]carbamoyl}pyrrolidine-2-carboxylate
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]propanamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}pyrrolidin-3-yl]methanol
1-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
4-ethyl-3-[1-(4-ethyl-5-methylthiophene-3-carbonyl)piperidin-3-yl]-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-6-(2-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-3-methylfuran-2-carboxamide
3-[2-(dimethylamino)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-8-[(3-methylphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(2R,3R)-1'-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
4-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1λ6-thiomorpholine-1,1-dione
2-[2-(dimethylamino)ethyl]-9-(3-hydroxy-4-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenoxy]pyridine
(4aS,7aR)-1-[(5-methylthiophen-2-yl)sulfonyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-(morpholin-4-yl)propyl]-3-(4-oxo-4H-chromen-6-yl)urea
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
methyl 7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-3-(quinoxalin-5-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate