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4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-(5-methyl-1,3,4-oxadiazol-2-yl)piperidin-4-ol
6-fluoro-4-methyl-2-{4-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]piperidin-1-yl}quinazoline
1-(5-chlorothiophene-2-carbonyl)-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
2-({[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]amino}methyl)-6-fluoroquinolin-4-ol
2-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyridine-4-carbonitrile
N-(3,4-difluorophenyl)-1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-3-amine
(2E)-3-(3,4-dimethoxyphenyl)-N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}prop-2-enamide
2-[5-(2,3-dimethoxyphenoxymethyl)-1,2,4-oxadiazol-3-yl]pyrazine
4-[(3-fluoro-5-methylphenyl)methyl]-1-(3-methoxyphenyl)piperazin-2-one
2-{[3-(2,5-dihydro-1H-pyrrole-1-carbonyl)phenyl]amino}acetic acid
1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(propan-2-yl)-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)spiro[2.3]hexane-1-carboxamide
3-[1-(2-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-5-methyl-1H-pyrazole
3-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]benzamide
1-[1-(3-phenylpropyl)-5-[1-(propan-2-yl)piperidin-4-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperidin-4-ol
1-(2,6-dimethoxypyridine-3-carbonyl)-3,4,4-trimethylpyrrolidin-3-ol
3-(2-amino-1,3-thiazol-4-yl)-1-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]propan-1-one
N2-[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-N1-(3-methylpyridin-4-yl)ethane-1,2-diamine
1-[5-(2-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]-3-propoxypiperidine
8-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N,N-diethyl-4-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}aniline
3-(4-hydroxyphenyl)-2-phenyl-N-{2-[(pyridin-3-yl)amino]ethyl}propanamide
{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
N-(3-chloro-4-fluorophenyl)-3-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}propanamide
N-cyclopropyl-3-{1-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]piperidin-4-yl}propanamide
1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
3-{2-[(3S,4S)-3-hydroxy-4-{[(3-methoxyphenyl)methyl](methyl)amino}pyrrolidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
methyl 6-{[methyl(propan-2-yl)amino]methyl}-3-(1,3-thiazole-5-amido)thieno[2,3-b]pyridine-2-carboxylate
2-{[(1-hydroxybutan-2-yl)[(2-methylphenyl)methyl]amino]methyl}-6-methylpyridin-3-ol
1-(2-aminoethyl)-N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(pyrrolidin-3-yl)benzamide
5-(3-chlorophenyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1,2,4-triazin-3-amine
3-[(4-fluorophenyl)methyl]-N-[2-(3-methoxyphenyl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
5-(3-benzoylpiperidine-1-carbonyl)-1,3-benzothiazole
(3R,4R)-1-[(5-chlorothiophen-2-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
2-[(3-methoxyphenyl)methyl]-4-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}morpholine
4-methoxy-N-(1-{1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
2-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{2-[5-(1,4-oxazepane-4-carbonyl)thiophen-2-yl]pyrrolidin-1-yl}-2-(propan-2-yloxy)ethan-1-one
methyl 1-[(3S,5S)-5-{[(4-methoxyphenyl)methyl]carbamoyl}-1-(3-methylbut-2-en-1-yl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-(5-benzyl-1,3,4-thiadiazol-2-yl)-3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carboxamide
1-(4,7-dimethylquinazolin-2-yl)-N-(1-methoxybutan-2-yl)piperidine-4-carboxamide
1-[(3,4-dimethylphenyl)methyl]-4-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperazin-2-one
1-[1-(benzenesulfonyl)piperidin-3-yl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(naphthalen-2-yl)acetamide
3-(2-fluorophenyl)-1-methyl-3-{2-oxo-2-[4-(pyridin-4-yl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
4-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-(quinolin-8-ylmethyl)piperidin-4-ol
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-5-methyl-1,3,4-oxadiazol-2-amine