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N-cyclopropyl-1-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-[2-(pyridin-3-yl)piperidin-1-yl]propan-1-one
3-{[3-(2-hydroxyethoxy)phenyl]methyl}-9-methoxy-N-methyl-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(azocan-1-yl)-3-(2-methoxy-5-{[(oxan-4-yl)amino]methyl}phenoxy)propan-2-ol
6-(benzylamino)-N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
6-hydroxy-4-propyl-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
N-[(2-propyl-1,3-thiazol-4-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
ethyl(methyl){[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}amine
N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-4-(2-methylpropyl)benzamide
(2S)-2-amino-1-{4-[3-(4-benzylpiperidin-1-yl)-3-oxopropyl]piperidin-1-yl}propan-1-one
1-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(1,2-oxazolidin-2-yl)propan-1-one
2-methyl-3-{[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}quinoxaline
5-(methoxymethyl)-N-[1-(5-{[(4-methoxyphenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]furan-2-carboxamide
1-benzyl-N-cyclopropyl-4-oxo-5-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1,4-dihydropyridine-3-carboxamide
N-(2-methoxyethyl)-1-{1-[2-(2H-1,2,3,4-tetrazol-2-yl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
(1-{[5-(2-methoxypyrimidin-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}cyclobutyl)methanol
5-ethyl-3-[2-(4-methoxyphenyl)ethyl]-5-{1-[1-(pyridin-2-yl)propan-2-yl]piperidin-4-yl}imidazolidine-2,4-dione
5-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-2-methoxypyridine
1-(cyclobutylmethyl)-4-[(3,4,5-trimethoxyphenyl)methyl]piperazine
1-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-3-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
3-ethyl-6-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-3H-imidazo[4,5-b]pyridin-2-amine
1-{1-[(dimethyl-1,3-thiazol-2-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
(3aR,6aR)-N,2-dimethyl-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-(carbamoylamino)-N-[(3R,4S)-1-(5-chloro-3-fluoropyridin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
6-ethyl-N-methyl-N-(propan-2-yl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[(3,4,5-trifluorophenyl)methyl]piperidine
[(5-methyl-1,2,4-oxadiazol-3-yl)methyl](propan-2-yl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
1-[1-(4-ethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(methylsulfanyl)ethan-1-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3,4,5-trimethoxy-N-methylbenzamide
2-(pyridin-4-yl)-N-[(4-sulfamoylphenyl)methyl]pyrimidine-5-carboxamide
N-{[7-(2-cyclohexylacetyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}furan-2-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}acetamide
N-(but-2-yn-1-yl)-4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(furan-2-ylmethyl)benzamide
6-[1-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)piperidin-3-yl]pyrimidin-4-ol
4-(1-ethyl-1H-imidazol-5-yl)-3-methyl-4H,5H,6H,7H-[1,2]thiazolo[5,4-b]pyridin-6-one
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-1-(2-phenylethyl)piperidine-3-carboxamide
[4-({1-[(5-ethylfuran-2-yl)methyl]pyrrolidin-3-yl}methyl)phenyl]methanol
9-(cyclopropylmethyl)-4-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-cyclohexyl-N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methyl-1H-pyrazole-4-carboxamide
6-fluoro-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1H-indazole
2-[1-(pyrimidin-4-yl)azetidin-3-yl]-1H-1,3-benzodiazole
1,5-dimethyl-4-({methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)urea
N-({3-methyl-7-[2-(1H-pyrazol-1-yl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
5-(2-methylpropyl)-3-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-1,2-oxazole
4-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-1,4-oxazepan-6-ol
N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyridin-4-amine
3-(3-chlorophenyl)-N-methyl-N-(oxan-4-yl)-3-phenylpropanamide