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1-[5-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]butan-2-ol
3-({4-[1-(2,5-dimethylfuran-3-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)pyridine
2-{3-methoxy-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-1H-1,3-benzodiazole
N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-4-(pyridin-3-yl)pyrimidin-2-amine
3,3-dimethyl-4-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperazin-2-one
3-benzyl-8-(cyclohex-3-en-1-ylmethyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{1-[(3,4-dimethylphenyl)methyl]piperidin-4-yl}-3-[(4-fluorophenyl)methyl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
8-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
methyl[(1-propyl-1H-imidazol-2-yl)methyl][1-(pyridin-4-yl)ethyl]amine
N-(1-{7-[(3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1-methylpiperidine-4-carboxamide
2-amino-6-[4-(difluoromethoxy)phenyl]-4-(pyridin-3-yl)pyridine-3-carbonitrile
N-{7-oxo-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl}pyridine-3-carboxamide
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]pentane-1,2-dione
1-phenyl-4-[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-3-yl]piperazine
1-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-2-[(4-methoxyphenyl)methyl]-1H-1,3-benzodiazole
N-[(7-{[4-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-2-phenoxyacetamide
5-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-(oxolan-3-yl)-1,2-oxazole-3-carboxamide
1-(2,3-difluoro-6-methoxybenzoyl)-4-[(2-fluorophenyl)methyl]-1,4-diazepane
[4-(2-phenoxyethyl)-1-(pyridin-3-ylmethyl)piperidin-4-yl]methanol
4-chloro-2-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-1H-indole
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-[2-(3-fluorophenyl)ethyl]-1-[(2-fluorophenyl)methyl]pyrrolidine-2-carboxamide
N-[2-(2-methoxyphenyl)ethyl]-2-[4-(4-{[1-(1,3-thiazol-5-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]acetamide
N-[(5-{1-[3-(pyridin-3-yl)propyl]-1H-pyrazol-3-yl}furan-2-yl)methyl]cyclopent-3-en-1-amine
N-[1-(2,5-difluorophenyl)cyclopropyl]-3-(1-methyl-1H-pyrazol-4-yl)propanamide
3-[1-(6-aminopyridine-2-carbonyl)piperidin-4-yl]-N-benzyl-N-methylpropanamide
N-{[6-chloro-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}benzenesulfonamide
N-(1-{2-[3-(carbamoylmethyl)-1-ethyl-1H-1,2,4-triazol-5-yl]-1H-indol-3-yl}propan-2-yl)acetamide
2-cyclopentyl-N-[3-(4-{[(2,3-dimethoxyphenyl)methyl]amino}piperidin-1-yl)phenyl]acetamide
(2S)-2-amino-3-(4-hydroxyphenyl)-1-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propan-1-one
3,5-difluoro-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyridine-2-carboxamide
N-[(2R,3R)-1'-(4-oxo-3,4-dihydrophthalazine-1-carbonyl)-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]cyclopropanecarboxamide
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-3-(1H-1,2,4-triazol-1-yl)adamantane-1-carboxamide
2-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
3-fluoro-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)benzamide
2-(2-aminoethyl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}quinazolin-4-amine
5-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-3-(1-methyl-1H-1,2,3-benzotriazol-5-yl)urea
(3aR,5S,6S,7aS)-2-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-isoindole-5,6-diol
4-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-N,N-dimethyl-4-oxobutanamide
2-(dimethylamino)-N-{[5-(3,6-dimethylpyrazin-2-yl)-7-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
3-(2-{[3-(2-hydroxyethoxy)phenyl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)phenol
1-(azocan-1-yl)-3-[2-methoxy-5-({[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
ethyl 5-[(5-acetamidothiophen-2-yl)methyl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-tert-butyl-3-[(3-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
(1S,5R)-N-(propan-2-yl)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
2-[(4aS,8aR)-1-(2-methylpropyl)-2-oxo-decahydro-1,6-naphthyridine-6-carbonyl]benzonitrile
(2S,4S,5R)-5-(2,3-difluorophenyl)-4-(4-hydroxypiperidine-1-carbonyl)-1-methylpyrrolidine-2-carboxylic acid
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-[3-(oxolan-2-yl)propyl]benzamide