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3-chloro-N-[(4-methoxyphenyl)methyl]-N-(3-methoxypropyl)-1H-indole-2-carboxamide
5-(2-methoxyacetamido)-N-methyl-N-(2-methylpropyl)-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
5-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-1,2,3-benzotriazole
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-[(3,4-dimethoxyphenyl)methyl]piperazin-2-one
4-hydroxy-2-(phenoxymethyl)-N-[2-(pyridin-4-yl)ethyl]pyrimidine-5-carboxamide
N-{[1-(carbamoylmethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}-N-(prop-2-en-1-yl)morpholine-4-carboxamide
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-N-(2-hydroxyethyl)pyridine-2-carboxamide
ethyl 2-{2-[3-(3-methoxyphenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-methylacetamido}acetate
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-(propan-2-yl)piperidin-4-amine
2-{1-[(4-ethoxyphenyl)methyl]-4-(isoquinolin-5-ylmethyl)piperazin-2-yl}ethan-1-ol
5-[(2-fluorophenyl)methyl]-5-[1-(2-phenylpropanoyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
N-ethyl-2-[2-(hydroxymethyl)phenyl]pyridine-4-carboxamide
2-cyclopropyl-4-methyl-N-[2-(2-methylpropanesulfonyl)ethyl]pyrimidine-5-carboxamide
3-(2-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)phenol
2-[(6-hydroxy-1,4-oxazepan-4-yl)methyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
4-(furan-2-carbonyl)-9-methoxy-7-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(5-methoxy-1H-indol-2-yl)methyl]-3-azaspiro[5.5]undecan-9-amine
2-cyclobutanecarbonyl-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
4-[2-(2-cyclohexyl-1H-imidazol-1-yl)-1-(pyridin-3-yl)ethyl]morpholine
3-(3-{[2-(dimethylamino)ethyl](methyl)amino}piperidine-1-carbonyl)-2-methyl-4,5,6,7-tetrahydro-1-benzofuran-4-one
2-(8-{[5-(4-chlorophenyl)furan-2-yl]methyl}-1-ethyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl)acetamide
methyl (3aS,6aS)-2-[(3E)-hex-3-enoyl]-5-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylate
(2E)-N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-3-(4-methoxyphenyl)prop-2-enamide
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
N-methyl-N-(oxan-4-yl)-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[(2,3,4-trifluorophenyl)methyl]pyrrolidin-3-yl]acetamide
N-methyl-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[2-(oxan-4-yl)ethyl]-1,2-oxazole-3-carboxamide
N,2,6-trimethyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]quinoline-4-carboxamide
2-(2-{3-[1-(dimethylamino)ethyl]phenyl}-4-methylphenoxy)acetamide
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-5-(methoxymethyl)thiophene-2-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2-methoxy-2-methylpropyl)acetamide
(1R,5R)-3-cyclobutanecarbonyl-6-(1H-indol-5-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
methyl 1-({4-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-4-carboxylate
3-{[(4aS,8aR)-1-[3-(methylsulfanyl)propyl]-2-oxo-decahydro-1,6-naphthyridin-6-yl]methyl}benzonitrile
5-[2,5-dimethoxy-4-(methylsulfanyl)phenyl]-3-methyl-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
3-{[4-(hydroxymethyl)oxan-4-yl]methyl}-3-methyl-1-[4-(1H-pyrazol-1-yl)phenyl]urea
N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]propanamide
2-(cyclopropylmethyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-{2-[1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]{[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
1-(piperidin-1-yl)-3-(4-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}phenoxy)propan-2-ol
9-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
3-{3-[(3,4-dimethylphenyl)amino]piperidine-1-carbonyl}-4H-pyrido[1,2-a]pyrimidin-4-one
5-methoxy-4-oxo-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1,4-dihydropyridine-2-carboxamide
2-(5-ethyl-1,3-oxazole-4-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
N-cyclopropyl-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-(pyridin-2-ylmethyl)acetamide
1-[6-hydroxy-4-(1,3-thiazol-4-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
ethyl (4aS,8aR)-6-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]-decahydro-1,6-naphthyridine-4a-carboxylate