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3-phenoxy-N-{[7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
methyl 3-(2-methylbutyl)-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[2-(trifluoromethyl)phenyl]urea
N-[2-(4-fluorophenyl)ethyl]-N-{[2-(3-hydroxypiperidin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}acetamide
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N,N-dimethylacetamide
N-({7-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)oxane-4-carboxamide
4-{[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]methyl}benzonitrile
4-phenyl-1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}azepane
1-{3-[4-(3,4-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
3-(4-chloro-1H-pyrazol-1-yl)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-(4-methoxyphenyl)-4-[1-(pyridin-2-ylmethyl)piperidin-3-yl]piperazine
1-[4-(benzyloxy)piperidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
(1R,5R)-3-(2-benzyl-1,3-thiazole-4-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(1H-pyrrol-2-yl)-4-(3,3,3-trifluoropropyl)pyrimidine
3-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}pyridin-2-amine
3-(2-fluorophenyl)-6-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)-1-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazine
N,15-dimethyl-13-oxo-9-(pyridin-3-yl)-4-(trifluoromethyl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
5-{2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}thiophene-2-carboxylic acid
1-({4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-3-carboxamide
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
N-{[1-(1H-indol-3-ylmethyl)piperidin-3-yl]methyl}-1H-indazole-3-carboxamide
7-(3-chloro-4-fluoro-1-benzothiophene-2-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
(4aR,7aS)-1-benzyl-4-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{4-benzyl-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
3-(3-methoxyphenyl)-N-(4,4,4-trifluorobutyl)-1H-pyrazole-5-carboxamide
1-{4-[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
N,N-diethyl-1-(1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
5-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]pyridin-2-ol
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-3-(pyridin-4-yl)propan-1-one
2-(1-ethyl-1H-pyrazole-4-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
3-(3-phenyl-1,2,4-thiadiazol-5-yl)-1-(pyridin-2-ylmethyl)urea
6-(2-propyl-1H-imidazol-1-yl)pyridin-2-amine
1-benzoyl-N-phenylpiperidin-3-amine
2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
methyl({[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
2-(3-chlorophenoxy)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
9-{2-[4-(dimethylamino)phenyl]acetyl}-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-{2-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
3-{2-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}-3-(3-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
1-(cyclohexylmethyl)-3-hydroxy-3-{[methyl(2-methylpropyl)amino]methyl}piperidin-2-one
({3-[2-(4-cyclopropanecarbonylpiperazin-1-yl)ethoxy]phenyl}methyl)(methyl)(naphthalen-1-ylmethyl)amine
8-(4-hydroxybenzoyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
(3R,5S)-N3-(4-fluorophenyl)-1-[(4-hydroxyphenyl)methyl]-N5-[(4-methylphenyl)methyl]piperidine-3,5-dicarboxamide
5-[4-(methoxymethyl)piperidine-1-carbonyl]-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-2-one
2-[(3S,4S)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-7-methyl-4H-chromen-4-one
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-methyl-N-[3-(piperidin-1-yl)propyl]-1H-1,3-benzodiazole-7-carboxamide
1-cyclobutyl-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
5-(5-acetylthiophene-3-carbonyl)-N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(2-phenylethyl)-5-[3-(1H-pyrazol-4-yl)propyl]-1H-1,2,4-triazole