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5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-3-(5-methylfuran-2-yl)-1H-pyrazole
3-{2-[4-(adamantan-2-yl)piperazin-1-yl]-2-oxoethyl}-4-methylpiperazin-2-one
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-8-fluoro-N-methylquinoline-2-carboxamide
2-{2,8-diazaspiro[4.5]decan-2-ylmethyl}quinolin-8-ol
N-(2,4-dimethylphenyl)-3-[2-(2-hydroxyethyl)piperidin-1-yl]-3-oxopropanamide
1-[(diethylcarbamoyl)methyl]-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperidine
N-[(2-chlorophenyl)methyl]-3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]propanamide
3-benzoyl-1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidine
3-(3-hydroxyphenyl)-3-(4-hydroxyphenyl)-1-(1,2-oxazolidin-2-yl)propan-1-one
N,N-diethyl-1-({1-[2-(3-methoxyphenyl)acetyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
5-(2-methyl-1,3-benzoxazol-5-yl)-1,2,3,4-tetrahydroisoquinoline
(2S,4R)-1-[(4-chlorophenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)-N-(thiophen-2-ylmethyl)pyrrolidine-2-carboxamide
4-ethyl-3-[1-(2-methoxypyrimidine-5-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
3-[2-(3-fluorophenyl)ethyl]-1-(furan-2-carbonyl)piperidine
2-(2,3-difluorophenyl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}acetamide
N-(2-methyl-2H-1,2,3-triazol-4-yl)-5-{1-[2-(1H-1,2,4-triazol-1-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-{1-[1-(quinoxalin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}pyridine-3-carboxamide
1-(2-fluoro-6-methoxybenzoyl)-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
4-methyl-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-1,3-oxazole-5-carboxamide
N-tert-butyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-5-[(2-methylpropyl)amino]benzene-1-sulfonamide
3-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-1-[3-(methylsulfamoyl)phenyl]urea
N-methyl-2-(pyrrolidin-1-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-5,6,7,8-tetrahydroquinazoline-4-carboxamide
3-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-1-(pyrrolidin-1-yl)propan-1-one
(2S)-2-amino-N-[1-(4-fluorophenyl)-6-(propan-2-yloxy)-1H-indazol-3-yl]butanamide
3-{[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]sulfonyl}-N-[3-(methylsulfanyl)propyl]benzamide
6-[5-(2-chlorophenyl)furan-2-carbonyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
(1R,2R,6S,7S)-4-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-4-azatricyclo[5.2.1.02,6]decane
3-({1-cyclohexyl-3-[hydroxy(phenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)imidazolidine-2,4-dione
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
5,6-dimethoxy-2-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-1,2-dihydroisoquinolin-1-one
2-{4-[(8-fluoroquinolin-2-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-benzyl{[3-(3-methyl-2,5-dioxoimidazolidin-1-yl)phenyl]amino}sulfonamide
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
N-[(2-chloro-6-fluorophenyl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
6-[(3S,4R)-3-cyclopropyl-4-(oxane-4-amido)pyrrolidin-1-yl]pyridine-3-carboxylic acid
5-{1-[(2E)-3-(2-fluorophenyl)prop-2-enoyl]piperidin-4-yl}-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
methyl 6-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]pyrimidine-4-carboxylate
3-[5-(1-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidin-3-yl)-1,2,4-oxadiazol-3-yl]pyridine
4-tert-butyl-2-{[4-(1-methyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}phenol
1-(6-methyl-2H-1,3-benzodioxol-5-yl)-5-oxopyrrolidine-3-carboxylic acid
methyl 3-{[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]carbamoyl}benzoate
N-(1-{1-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
3,3-dimethyl-1-{[5-(quinolin-5-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}urea
2-{[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}-N-methylethane-1-sulfonamide
1-(4-benzylpiperazine-1-carbonyl)-6-(2-chloropyridine-4-carbonyl)-6-azaspiro[2.5]octane
4-(1H-imidazol-2-yl)-1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidine
(4aS,8aR)-6-(1H-1,2,3-benzotriazole-5-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
3-(2,3-dihydro-1H-inden-2-yl)-8-(1H-indol-2-ylmethyl)-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione