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5-(4-benzyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-methylfuran-2-carboxamide
N-ethyl-2-(4-methoxy-2-methylphenyl)pyridine-4-carboxamide
3-(2-{2-[2-(propylsulfanyl)pyrimidin-5-yl]-1H-imidazol-1-yl}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-acetyl-N-{[3-methyl-7-(4-methylbenzoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-3-carboxamide
N-(3-hydroxy-2,2-dimethylpropyl)-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
methyl N-({[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]carbamoyl}methyl)carbamate
1-ethyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1H-pyrazole-4-carboxamide
methyl 2-(3-{[(4-fluorophenyl)formamido]methyl}piperidine-1-carbonyl)benzoate
(2S)-4-methyl-2-[4-(pyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]pentanamide
5-[(2-chlorophenyl)methyl]-5-[1-(naphthalene-1-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
2-[2-methyl-4-oxo-1-(3-phenylpropyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]-N-(oxolan-3-yl)acetamide
9-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3-oxa-9-azaspiro[5.5]undecane
7-(cyclohexylmethyl)-2-(5-methylpyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-(2-phenylethyl)piperidin-2-one
N-(2-hydroxyethyl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
5-methoxy-2-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-4H-pyran-4-one
2-(2-{5-[2,5-dimethyl-1-(propan-2-yl)-1H-pyrrol-3-yl]-4-phenyl-1H-imidazol-1-yl}ethyl)pyrazine
2-{1-[(3,4-difluorophenyl)methyl]-4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl}ethan-1-ol
1-cyclopentyl-5-(furan-3-yl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
2-(4-methyl-1,4-diazepan-1-yl)-2-[6-(piperidin-1-yl)pyridin-3-yl]acetic acid
1-(4-fluorophenyl)-2,2-dimethyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)cyclopropane-1-carboxamide
ethyl 4-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}piperidine-1-carboxylate
4-({5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}amino)butan-1-ol
2-{[(adamantan-1-yl)carbamoyl]amino}-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetic acid
N-({1-[(2,3-difluorophenyl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}propanamide
N-[2-(2-chlorophenoxy)ethyl]-2-(phenylamino)pyrimidine-5-carboxamide
5-(3,5-dimethyl-1H-indole-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-methyl-1-[4-(morpholine-4-carbonyl)phenyl]urea
(3S,4S)-4-methyl-1-(1-methyl-1H-indole-3-carbonyl)piperidine-3,4-diol
1-(oxan-4-yl)-4-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}piperazine
N-[(2,4-difluorophenyl)methyl]-5-(2-methoxyphenoxymethyl)-1,2-oxazole-3-carboxamide
5-{1-[(3,4-difluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
(1R,5S)-6-[(2,3,4-trifluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-(2-methoxyethyl)-N-(thiophen-3-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-[2-(piperidin-1-yl)ethyl]-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
methyl 4-[5-(2,5-dihydro-1H-pyrrol-1-ylmethyl)-1,2,4-oxadiazol-3-yl]benzoate
2-[1-(dimethyl-1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]-1-methyl-1H-1,3-benzodiazole
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(1,3,4-thiadiazol-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(dimethylamino)-2-(4-methylphenyl)-N-(oxan-4-yl)acetamide
2-{4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperazin-1-yl}-1H-1,3-benzodiazole
5-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-1-methyl-1H-imidazole
3-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-6,7-dimethoxy-1,2-dihydroquinolin-2-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3,5-dimethyl-1,2-oxazole-4-carboxamide
2-(2-oxo-4-{2-[4-(propan-2-yl)morpholin-2-yl]acetyl}piperazin-1-yl)benzonitrile
N-ethyl-6-oxo-1-(pyridin-2-ylmethyl)-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
1-(3-chlorophenyl)-4-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperazin-2-one
2-{[5-(2-fluoro-6-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-5-methylpyrazine
(1-{[(4-cyclopentylpyrimidin-2-yl)(methyl)amino]methyl}cyclobutyl)methanol