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2-(1-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-3-oxopiperazin-2-yl)-N-methylacetamide
2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}({[4-(methylsulfanyl)phenyl]methyl})amino)ethan-1-ol
3-{1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]pyrrolidin-2-yl}pyridine
2-{4-[(4-fluorophenyl)methyl]-2,5-dioxo-4-(piperidin-4-yl)imidazolidin-1-yl}-N,N-dimethylacetamide
N-(1-benzyl-1H-pyrazol-3-yl)-2-(4-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-pyrazol-1-yl)acetamide
9-(3-methoxybenzenesulfonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
methyl 3-{[(3,5-dimethylphenyl)formamido]methyl}-5-[2-(1,3-thiazol-4-yl)acetamido]benzoate
4-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-1,4-diazepan-2-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]acetamide
1-cyclohexyl-4-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-2-one
1-[(2-fluoro-4-methoxyphenyl)methyl]-3-methoxypiperidine
1-[(4-chlorophenyl)methyl]-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-(3-methylphenoxy)ethan-1-one
ethyl 2-[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]-1,3-oxazole-4-carboxylate
6-(4-methoxyphenyl)-3-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2-dihydropyridin-2-one
1-(cyclohexylmethyl)-N3,N3-dimethyl-4-oxo-N5-{[4-(trifluoromethyl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
N-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(4-benzylpiperazin-1-yl)-3-[1-(6-methylpyridine-2-carbonyl)piperidin-3-yl]propan-1-one
1-[4-(adamantan-1-yl)piperazin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
6-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-N-(3-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
(2S,4S)-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-N-[2-(3-fluorophenyl)ethyl]-1-[(3-methylphenyl)methyl]pyrrolidine-2-carboxamide
4-[(2-chlorophenyl)methyl]-11-(morpholin-4-yl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-(3-{[2-(dimethylamino)ethyl](methyl)amino}piperidin-1-yl)-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
2-{4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-[(3-hydroxy-2,2-dimethylpropyl)amino]-N-(4-methylphenyl)propanamide
1-[3-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]pyrrolidin-2-one
N-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-3-(2-oxopiperidin-1-yl)propanamide
3-[2-amino-4-methyl-6-({[5-(methylcarbamoyl)furan-2-yl]methyl}amino)pyrimidin-5-yl]propanoic acid
N-benzyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-2-({3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}sulfanyl)acetamide
N-[3-(1H-1,2,4-triazol-1-yl)adamantan-1-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
6-(ethanesulfonyl)-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
3-[3-(4-fluorophenoxy)propyl]-5,5-dimethyl-1,3-oxazolidine-2,4-dione
1-[(2-methoxyphenyl)methyl]-N-[2-(3-methylpyridin-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
ethyl 1-{1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}piperidine-4-carboxylate
1-[1-(3-hydroxypropyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
methyl 5-[(2,3-dihydroxypropyl)amino]-3-(furan-2-amido)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2,5-dimethyl-4-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]pyrimidine
methyl 4-({[5-(4-chloro-2-methoxyphenoxymethyl)-1,2-oxazol-3-yl]formamido}methyl)benzoate
6-{[4-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-1,4-oxazepan-6-ol
1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
N,N-dimethyl-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-sulfonamide
6-[(2-hydroxy-3-methoxyphenyl)methyl]-N-[2-(2-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
4-methyl-1-{2-[2-(1-phenylethyl)-1H-imidazol-1-yl]ethyl}-1H-1,2,3-triazole
N-cyclopentyl-4-{4-[(furan-2-ylmethyl)(prop-2-yn-1-yl)amino]piperidin-1-yl}benzamide
3-{N-benzyl-1-[4-(piperidin-3-yl)phenyl]formamido}propanamide
N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-phenylbutanamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-(quinolin-6-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1-{7-[(4-methoxy-2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
(1R,5S)-3-[2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carbonyl]-3,8-diazabicyclo[3.2.1]octane