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methyl (2S)-2-{[3-(naphthalen-1-ylmethyl)-1,2-oxazol-5-yl]formamido}-3-phenylpropanoate
ethyl 4-(oxan-2-ylmethyl)-1-(phenylcarbamoyl)piperidine-4-carboxylate
N-[2-(3-methoxyphenyl)-1-[1-(3-phenylpropanoyl)piperidin-4-yl]ethyl]-N-methylthiophene-3-carboxamide
1-(3-chlorophenyl)-5-methyl-4-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]piperazin-2-one
ethyl 1-{2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl}-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
3-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-1-[2-(morpholin-4-ylmethyl)phenyl]urea
7-[2-(pyridin-3-yl)piperidine-1-carbonyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
4-(1H-imidazol-1-ylmethyl)-1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine
2-{[4-(2,5-dimethylphenyl)piperazin-1-yl]methyl}-6-methylquinazolin-4-amine
2-phenoxy-1-(4-{5-[(1E)-prop-1-en-1-yl]-2-(pyridin-3-yl)pyrimidin-4-yl}piperidin-1-yl)propan-1-one
N-cyclooctyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-[1-(2-carbamoylethyl)-1H-pyrazol-4-yl]-N,N-diethylbenzamide
3-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]quinoline
4-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-6-[(5-methyl-1,2,4-oxadiazol-3-yl)methoxy]-1-(propan-2-yl)-1,4-diazepan-2-one
[(4-fluorophenyl)methyl]({[5-(1H-pyrazol-5-yl)furan-2-yl]methyl})(pyridin-4-ylmethyl)amine
3-(3-hydroxy-3-methylbutyl)-N-[3-(morpholin-4-yl)-3-oxopropyl]benzamide
1-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-[3-(pyridin-4-yl)azetidine-1-carbonyl]quinoline
N-[(3S,4R)-1-[(1-benzyl-1H-imidazol-5-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
(2S,4S)-4-[4-(3,5-difluorophenyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxylic acid
5-ethyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
cyclohexyl({4-[(2,3-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl})methanol
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2,4-dimethoxy-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzamide
3-[(1-benzylpiperidin-4-yl)oxy]-N-[2-(dimethylamino)ethyl]-4-methoxybenzamide
3-(2-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
(cyclopropylmethyl)(2-methoxyethyl){[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
(4aR,7aS)-4-(4-fluoro-3-methylbenzoyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-(3-methoxyphenyl)-4-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]-1H-pyrazole
5-(8-methoxyquinolin-5-yl)pyrimidin-2-amine
1-ethyl-3-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]piperidine-3-carboxamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)ethan-1-one
5-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-1-ethyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
[1-(1,2,3,4-tetrahydronaphthalen-2-yl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
(2R)-2-[5-(5-cyano-1-methyl-1H-pyrrol-3-yl)-4-phenyl-1H-imidazol-1-yl]-3-hydroxypropanoic acid
2,4-dimethyl-N-{[7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
2-(4-chlorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-1-phenyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
1-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-4-(pyridin-3-yl)piperazine
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)cyclopropanecarboxamide
6-[(3-fluorophenyl)methyl]-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
3-[(cyclopropylmethyl)amino]-5-(dimethylsulfamoyl)-N-methyl-N-[1-(pyridin-2-yl)ethyl]benzamide
2-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)-4-(pyrazin-2-yl)phenol
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanamide
1-[5-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-2-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
2-[(6-hydroxy-1,4-oxazepan-4-yl)methyl]-6,8-dimethylquinolin-4-ol
5-{[3-(piperidin-1-ylmethyl)piperidin-1-yl]methyl}-2-(thiophen-2-yl)pyrimidine
1-[(3-chlorophenyl)methyl]-4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(1-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-6-azaspiro[2.5]octan-6-yl)-2-(2-methylphenyl)ethan-1-one