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1-({1-[1-(4-methylpentan-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)piperidin-4-ol
2-ethyl-N-{2-[2-(trifluoromethoxy)phenyl]ethyl}pyrimidine-5-carboxamide
N,8-dimethyl-3-{[methyl(pyridin-3-ylmethyl)amino]methyl}-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
N-methyl-N-(1-methylpiperidin-4-yl)-3-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-3-yl)propanamide
{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}[1-(pyridin-2-yl)propan-2-yl]amine
1-(2,3-dihydro-1H-inden-5-yl)-3-ethyl-5-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepin-9-yl}-1H-1,2,4-triazole
1-{3-[5-(2-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl}-2-(pyridin-4-ylsulfanyl)ethan-1-one
1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
5-ethyl-2,3-dimethyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-{[(1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperidin-3-yl)oxy]methyl}pyridine
N-[1-(2,4-dimethylphenyl)ethyl]-3-acetamidobenzamide
5-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(3-fluoro-4-methoxybenzoyl)piperidine
(3R,5S)-1-benzyl-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[2-(1H-imidazol-4-yl)ethyl]piperidine-3,5-dicarboxamide
9-[(2-ethylphenyl)methyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[2-(benzyloxy)ethyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-2-methoxyethan-1-one
3-{2-[2-(3-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)ethyl]piperidine-1-carbonyl}-1,2,5,6,7,8-hexahydroquinolin-2-one
dimethyl(2-{2-[1-(pyrrolidine-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
2-(dimethylamino)-7-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
N-({1-[(3-chloropyridin-4-yl)methyl]piperidin-3-yl}methyl)-2,2-dimethylpropanamide
N-methyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}-N-[(1-phenylpyrrolidin-3-yl)methyl]acetamide
(3aR,6aS)-5-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(pyridin-2-yl)-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}-N-[1-(propan-2-yl)-1H-1,2,4-triazol-5-yl]benzamide
methyl 1-({4-[5-(methoxymethyl)thiophene-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-4-carboxylate
4-{3-[(3,4-dimethoxyphenyl)amino]piperidine-1-carbonyl}-1,2-dihydrophthalazin-1-one
1-(2-methoxyphenyl)-5-[(2R)-oxolan-2-yl]-3-(2-phenylethyl)-1H-1,2,4-triazole
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-(1H-pyrrol-1-yl)propanamide
4-(4-{4-[2-(dimethylamino)ethoxy]piperidine-1-carbonyl}phenyl)-2-methylbutan-2-ol
N-[(2R,3R)-2-methoxy-1'-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
2-(1H-imidazol-1-yl)-N-{[3-methyl-7-(2,3,6-trifluorobenzoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}acetamide
7-cyclohexyl-2-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-(4-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazin-1-yl)pyrazine-2-carbonitrile
(1R,5R)-3-benzoyl-6-[(1-methyl-1H-indol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}-1-methyl-3-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
ethyl[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl](1H-indol-4-ylmethyl)amine
4-[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]phenol
2-(dimethylamino)-2-(4-fluorophenyl)-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
N-[2-(3-methoxyphenyl)-1-{1-[2-(2-methylphenyl)acetyl]piperidin-4-yl}ethyl]-N-methylpyridine-3-carboxamide
N3-butyl-N5-[1-(4-fluorophenyl)ethyl]-1-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-{[4-(3-methoxyphenyl)piperazin-1-yl]methyl}-1,6-dimethyl-1,2-dihydroquinolin-2-one
1-(3-fluoropyridin-2-yl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylic acid
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-(quinolin-5-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3-{[methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenyl)ethan-1-one
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
1-(cyclohexylmethyl)-N-[2-(4-fluorophenoxy)ethyl]-6-oxopiperidine-3-carboxamide
(2E)-N-methyl-3-(1-methyl-1H-pyrazol-4-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]prop-2-enamide
(benzylsulfamoyl)[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]amine
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-4,4,4-trifluorobutanamide