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1-(2-amino-5-ethylpyrimidin-4-yl)-4-methylazepan-4-ol
2-methyl-4-[4-(2-methylpyrrolidine-1-carbonyl)phenyl]butan-2-ol
(1S,4S)-2-[5-(2,4-difluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-2-azabicyclo[2.2.1]heptane
4-methyl-14-[2-(pyrrolidin-1-yl)pyrimidin-5-yl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-[3-(1H-imidazol-1-yl)propyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
4-(morpholine-4-sulfonyl)-2-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]phenol
3-hydroxy-2-[5-(3-hydroxy-4-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]propanoic acid
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-5,7-dimethylpyrazolo[1,5-a]pyrimidine
2-(1H-imidazol-1-yl)-1-{3-[2-(4-methyl-1,4-diazepan-1-yl)-2-oxoethyl]morpholin-4-yl}ethan-1-one
5-ethyl-1'-(2-methoxypyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)hex-5-ynamide
N-[2-(4-fluorophenoxy)ethyl]-6-methyl-2-oxo-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-cyclopropanecarbonyl-4-{4-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]phenoxy}piperidine
1-[2-(3,3-diphenylpiperidin-1-yl)ethyl]pyrrolidin-2-one
1-propyl-4-[3-(1H-pyrazol-1-yl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-{5-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
2-butyl-8-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(4-chlorophenyl)-3-[1-(cyclopropanesulfonyl)piperidin-3-yl]propanamide
3,4,5-trimethoxy-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}benzamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]benzamide
N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carboxamide
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-methyl-N-[(3-methylpyridin-4-yl)methyl]pyridin-2-amine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-propyl-1,3-thiazole-4-carboxamide
5-[1-(3-methylphenyl)-1H-imidazol-2-yl]-2-(pyridin-2-yl)pyrimidine
3-({2-[1-(2-ethoxybenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(2-fluorobenzoyl)piperidin-4-yl]oxy}benzamide
3-fluoro-5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}pyridine
3-(but-2-yn-1-yl)-5-[1-(3-phenoxypropanoyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
4-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[4-(4-methoxybutyl)piperazin-1-yl]pyrimidine
(2E)-3-(2-chlorophenyl)-1-(3-{5-methyl-2-[(pyridin-2-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)prop-2-en-1-one
1-(2-{methyl[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)piperidin-2-one
1-(1-benzylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
1-methyl-2-oxo-8-(1H-pyrazole-3-carbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-methyl-4-{4-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]butan-2-yl}piperazine
5-ethyl-2-{1-[2-(pyridin-3-yloxy)propyl]-1H-imidazol-2-yl}pyridine
[2-(diethylamino)ethyl]({[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl})ethylamine
N-[(2-{2-[(dimethylsulfamoyl)amino]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-2,3-dimethyl-1H-indole-7-carboxamide
1-(3-methoxyphenyl)-5-methyl-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperazin-2-one
N-[(3-chlorophenyl)methyl]-2-[1-cyclopentyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
2-{4-phenyl-5-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-1-yl}-1-(pyridin-3-yl)ethan-1-ol
2-[4-(3,6-dimethylpyrazin-2-yl)-1H-pyrazol-1-yl]-N-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]acetamide
5-[(dimethylamino)methyl]-N-(furan-3-ylmethyl)-N-methylfuran-2-carboxamide
1-cyclopentyl-4-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]pyrrolidin-2-one
4-methyl-6-[4-(3,5,7-trimethyl-1H-indole-2-carbonyl)piperazin-1-yl]pyrimidin-2-amine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}propanamide
8-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
(3S,4R)-1-(6-ethyl-5-fluoropyrimidin-4-yl)-4-methylpiperidine-3,4-diol
8-cyclopropanecarbonyl-2-(2-phenylacetyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid