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2-cyclopentyl-N-(3-methoxypropyl)-N-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}acetamide
N-{[7-(2-ethylbutanoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-2-sulfonamide
2-amino-6-(7-methoxy-1-benzofuran-2-yl)-4-(piperidin-4-yl)pyridine-3-carbonitrile
4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-(4-methoxyphenyl)-2,2-dimethylpiperazine
1-[2-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
1-(3-methoxypropyl)-8-[(4-methylphenyl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]acetamide
3-methyl-N-{[5-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
N-({8-[(2,4-dimethoxy-3-methylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-methoxyacetamide
(2S)-2-[2-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamido]-3-methylbutanamide
2-{5-[2-(3-chloro-1,2-oxazol-5-yl)ethyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}-6-methylpyridine
3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]benzamide
4-(2,6-dimethylpyridin-3-yl)-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methylpyrimidin-2-amine
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-methyl-2-phenyl-N-(piperidin-4-yl)acetamide
8-methyl-3-[1-(pyridin-3-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
N-[(2R,3R)-1'-(cyclopent-1-ene-1-carbonyl)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-methyl-N-(2-phenoxyethyl)acetamide
propyl(pyridin-3-ylmethyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
4-(1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-4-yl)-6-(pyrrolidin-1-yl)pyrimidine
2-(4-{[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[1-(2-phenyl-1,3-thiazol-5-yl)ethyl]propanamide
2-methyl-4-{3-[(2S)-2-(morpholine-4-carbonyl)pyrrolidine-1-carbonyl]phenyl}butan-2-ol
1-ethyl-8-{[4-(methylsulfanyl)phenyl]methyl}-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-methyl-1-[4-(2-phenylethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]butan-1-ol
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(2,6-dimethoxypyrimidin-4-yl)piperazin-2-one
N-cyclopentyl-3-{5-[(1-methyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
7-[2-(4-phenylphenyl)acetyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
4-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1λ6-thiomorpholine-1,1-dione
N-[3-(methylsulfanyl)phenyl]-3-[(3S,4R)-1-(pyridin-2-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
1-[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(pyrazin-2-yl)propan-1-one
2-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-7-methyl-4H-chromen-4-one
N-[2-methyl-2-(morpholin-4-yl)propyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylpyrazine-2-carboxamide
N-butyl-4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxybenzamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(pyridin-3-ylmethyl)thiophene-3-carboxamide
methyl 4-{4-[4-(1H-pyrazol-1-yl)butanoyl]piperazin-1-yl}benzoate
3-[(2R,3R,6R)-5-(2,4-difluorobenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
6-[3-chloro-5-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyrazine-2-carboxamide
N-[7-(4-benzylpiperazine-1-carbonyl)-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazol-5-yl]-2-methoxyacetamide
N-{2-[4-(2,2-dimethylpropyl)morpholin-2-yl]ethyl}cyclobutanecarboxamide
N-[3-(morpholin-4-yl)propyl]-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-3-methyl-1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]urea
1-(carbamoylmethyl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methylpiperidine-4-carboxamide
3-[(3R,4S)-1-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]piperidine-4-carboxamide
methyl 3-benzamido-5-[(3-methylbutyl)amino]-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
methyl (2S,4R)-4-(1-hydroxynaphthalene-2-amido)-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
N-[(2-methyl-1H-indol-5-yl)methyl]-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide