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4-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]-1-methyl-1,2-dihydroquinolin-2-one
N-(2-methylpropyl)-5-oxo-1-(pyridin-4-ylmethyl)-N-(thiophen-3-ylmethyl)pyrrolidine-3-carboxamide
1-(furan-2-ylmethyl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperazine
N-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
N-[(4-methoxyphenyl)methyl]-N-(oxolan-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-(cyclohex-3-en-1-ylmethyl)-3-[4-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,6-dimethylimidazo[1,2-a]pyridine-2-carboxamide
8-[(4-chlorophenyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(3-methyl-4-{[3-(pyrrolidine-1-carbonyl)piperazin-1-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
4-[(dimethylamino)methyl]-N-[(8-methoxyquinolin-5-yl)methyl]-N-methylbenzamide
6-{2-cyclopropyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-2-carbonitrile
4-(2,4-dimethyl-1,4-diazepane-1-carbonyl)-2-(1-ethyl-1H-pyrazol-4-yl)quinoline
2-butyl-8-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
3-(1-ethyl-1H-1,2,4-triazol-3-yl)-1-methyl-1-[(2-methylphenyl)methyl]urea
4-{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-[(3-methylphenyl)methyl]piperazin-2-one
N-benzyl-5-{[4-(diethylamino)phenyl]methyl}-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(4-carbamoylphenyl)-4-methoxybenzoic acid
3-(1H-1,3-benzodiazol-2-yl)-1-{4-[3-(morpholin-4-yl)-3-oxopropyl]piperidin-1-yl}propan-1-one
3-{imidazo[1,2-a]pyridin-2-yl}-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)propanamide
3-(2,3-dihydro-1H-inden-2-yl)-8-{[5-(methoxymethyl)furan-2-yl]methyl}-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N5-[2-(cyclohex-1-en-1-yl)ethyl]-N3-ethyl-1-[(2-methoxyphenyl)methyl]-N3-(2-methylprop-2-en-1-yl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(3S,4R)-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
ethyl 5-(naphthalene-1-carbonyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
5-(2,6-dimethoxyphenyl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1,2,4-triazin-3-amine
(2E)-N-({3-methyl-7-[3-(prop-2-en-1-yloxy)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide
3-[3-(dimethylamino)propyl]-5-{1-[(2E)-4-methylpent-2-enoyl]piperidin-4-yl}-5-[(2-methylphenyl)methyl]imidazolidine-2,4-dione
1-benzyl-N-[2-(ethanesulfonyl)ethyl]-1H-pyrazole-4-carboxamide
3-butyl-1-methyl-4-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperazin-2-one
6-[(4-chlorophenyl)amino]-1-(2-methylprop-2-en-1-yl)-1H,4H,5H,8H-imidazo[4,5-e][1,3]diazepine-4,8-dione
N-(3,3-diphenylpropyl)-6-(4-methyl-1H-imidazole-2-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
8-[(2E)-3-phenylprop-2-en-1-yl]-1-oxa-8-azaspiro[4.6]undecan-9-one
(1S,5R)-6-(cyclopropylmethyl)-3-(1H-indol-5-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[(4-methoxypyridin-2-yl)methyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[1-(thiophen-3-yl)propan-2-yl]acetamide
(1R,5S,6S)-N-[1-(3-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[4-(pyridin-3-ylmethyl)piperazin-1-yl]propan-1-one
4-(1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)morpholine
2-chloro-N-{2-[(1-ethyl-5-oxopyrrolidin-3-yl)formamido]ethyl}benzamide
(2E)-3-(3,4-difluorophenyl)-N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)prop-2-enamide
N-{1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-2-(2-fluorophenyl)ethyl}-N-methyl-3-(methylsulfanyl)propanamide
6-[(cyclopropylmethyl)amino]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
4-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidine
3-{[1-tert-butyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-7-fluoro-2-methyl-1H-indole
3-methoxy-6-(3-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyridazine
N-ethyl-5-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}pyrimidin-2-amine
[(3-{2-[4-(2-fluorobenzenesulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(thiophen-2-ylmethyl)amine
2-(3-acetyl-1H-indol-1-yl)-1-(2,5-dihydro-1H-pyrrol-1-yl)butan-1-one
2-amino-2-methyl-1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
4-{[(2,2-dimethyloxan-4-yl)(ethyl)amino]methyl}-1H-pyrazole-3-carboxylic acid
1-(2,3-dihydro-1H-inden-2-yl)-4-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperazine