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N-cyclopentyl-2-[methyl({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl})amino]propanamide
6-{9-oxo-8-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-3-carbonitrile
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2H-1,3-benzodioxole-5-carboxamide
2-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}-6-methoxyphenol
2-(dimethyl-1,2-oxazol-4-yl)-N-{[4-(oxolan-2-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)acetamide
1-[3-(4-fluorophenyl)benzoyl]-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
3-[2-oxo-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-4-(pyridin-3-ylmethyl)piperazin-2-one
N,N-dimethyl-2-({2-methyl-3-[(pyridin-3-ylmethyl)amino]phenyl}formamido)-2-phenylacetamide
ethyl 4-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}piperidine-1-carboxylate
1-[2-oxo-2-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-1-oxaspiro[4.4]nonan-2-one
4-[(2-methyl-1,3-thiazol-4-yl)methyl]-N-(1-phenyl-1H-pyrazol-5-yl)piperazine-1-carboxamide
(3S,4S)-4-(morpholin-4-yl)-1-(pyridin-2-ylmethyl)pyrrolidin-3-ol
(3S,4S)-1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
N-(2-acetamidoethyl)-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
methyl 5-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]-3-(2-methoxyacetamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-{[4-(4-chlorophenyl)-4H-1,2,4-triazol-3-yl]methyl}phenol
N-[(5-methyl-2-{3-[2-(4-methylphenoxy)acetamido]phenyl}-1,3-oxazol-4-yl)methyl]butanamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-[(3,4,5-trifluorophenyl)methyl]acetamide
3-(4-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)propanamide
N-{4-methyl-2-[2-(pyrimidin-2-ylsulfanyl)acetamido]phenyl}pentanamide
4-[2-(methylsulfanyl)propyl]-1-[2-(pyrrolidin-1-yl)ethyl]-1H-1,2,3-triazole
3-benzyl-N-{2-[2-(trifluoromethyl)phenyl]ethyl}-1,2-oxazole-5-carboxamide
4-(1H-imidazol-1-yl)-N-(1-phenylbutyl)benzamide
8-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2-methoxyphenyl)-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]piperidin-4-amine
5-[(1,4-dithiepan-6-yl)amino]-4-methylpentane-1,4-diol
2-{4-[(3ar,6ar)-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]piperazin-1-yl}-1-(piperidin-1-yl)ethan-1-one
4-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}-N-[(2-fluorophenyl)methyl]piperidine-1-carboxamide
(3R)-N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-[(5-methylfuran-2-yl)methyl]-3-[2-oxo-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]piperazin-2-one
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(2-methoxyethoxy)piperidine
1-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]cyclopropane-1-carboxamide
4-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-N-(5-methylpyridin-3-yl)benzamide
N-(3-cyanothiophen-2-yl)-3-({methyl[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)benzamide
6-(cyclohexylamino)-1-[(2,5-dimethylphenyl)methyl]-1H,4H,5H,8H-imidazo[4,5-e][1,3]diazepine-4,8-dione
1-cyclopropyl-3-(4-methoxyphenyl)-3-[2-oxo-2-(4-phenylpiperidin-1-yl)ethyl]pyrrolidine-2,5-dione
4-methyl-2-(4-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}piperidin-1-yl)-6-(propan-2-yl)quinazoline
5-{[2-(3,4-dichlorophenyl)morpholin-4-yl]methyl}-N-methylfuran-2-carboxamide
4-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-3-yl)benzoic acid
methyl 4-{[(2-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-5-oxopyrrolidin-2-yl}ethyl)amino]methyl}benzoate
4-(4-methyl-3-phenylpiperazine-1-carbonyl)pyridin-3-ol
3-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-1-cyclopropyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
1-[(4-methoxyphenyl)methyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-({7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}methyl)benzoic acid
N-(1-{4-[(2-fluoro-4,5-dimethoxyphenyl)methyl]phenyl}ethyl)acetamide
4-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonane-7-carbonyl]-6-(2-methylpropyl)-1,2-dihydropyrimidin-2-one
N'1-[1-(cyclohexylmethyl)piperidin-3-yl]cyclopropane-1,1-dicarboxamide
7-(cyclopropylmethyl)-2-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
7-fluoro-3-({[(3-methoxyphenyl)methyl](methyl)amino}methyl)-1,2-dihydroquinolin-2-one