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5-[1-(3-chlorobenzoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
2-(dimethyl-1,3-thiazol-5-yl)-N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}acetamide
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-4-(4-methylphenoxy)piperidine-4-carboxamide
1-[(2S)-2-amino-2-phenylacetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(2-ethoxypyridin-3-yl)methyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
2-methoxy-N-{3-[2-(5-oxopyrrolidin-2-yl)acetamido]phenyl}benzamide
3-(2-methoxyphenyl)-1-(7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
1-(4-fluorophenyl)-3-(2-methylpropyl)-5-(oxolan-2-yl)-1H-1,2,4-triazole
methyl 3-[(2-phenoxyacetamido)methyl]-5-[2-(1H-pyrazol-1-yl)acetamido]benzoate
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethylacetamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-5-methylpyrazine-2-carboxamide
4-fluoro-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]benzamide
2-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-N-(pyridin-2-ylmethyl)acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
1-[5-(2-methoxy-4-methylphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(pyrrolidin-1-yl)piperidine
methyl 2-[(butan-2-yl)sulfamoyl]-6-[2-(2,6-difluorophenyl)acetyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-cyclopropyl-1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-(3-methoxypropyl)-1H-pyrazole-4-carboxamide
1-[2-(2-hydroxyethoxy)ethyl]-5-methyl-5-phenylpiperidin-2-one
2-(4-methoxyphenyl)-N-({1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]piperidin-3-yl}methyl)acetamide
7-chloro-1-methyl-2-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-indole
3-[(4-methoxyphenyl)methyl]-N-(2-methylpropyl)-1,2-oxazole-5-carboxamide
1-[(4-fluorophenyl)methyl]-N-[3-(1H-indazol-1-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
4-{1-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-2-yl}-2-phenyl-1,3-oxazole
8-(4-amino-3-hydroxybutanoyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-[(5-chlorothiophen-2-yl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
1-(4-{[(2R)-1-hydroxypropan-2-yl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
3-{[1-(3-cyanopyridin-2-yl)piperidin-4-yl]amino}-N-(1,3-thiazol-2-yl)propanamide
2-(2-chloro-4-fluorophenyl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(2S,4R)-N,N-diethyl-1-(4-hydroxybenzoyl)-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
1-(4-{[5-(4-fluorophenyl)-2-hydroxyphenyl]methyl}piperazin-1-yl)ethan-1-one
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
N,7-dimethyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1-benzofuran-2-carboxamide
(5S,9aS,9bS)-5-(3,4-difluorophenyl)-2-[(3-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(benzyloxy)-N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)acetamide
(1R,7S)-N-methyl-4-oxo-3-[2-(pyridin-4-yl)ethyl]-N-(pyrimidin-4-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(2S,4R)-N-(2-phenylethyl)-1-[(2E)-3-phenylprop-2-en-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
N-[(1-cyclopentylpiperidin-3-yl)methyl]-2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(piperidin-1-yl)ethyl]acetamide
5,6-dimethyl-2-oxo-N-[(4-phenylmorpholin-2-yl)methyl]-1,2-dihydropyridine-3-carboxamide
3-ethoxy-1-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
N-(2-phenylphenyl)-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carboxamide
N-{[4-(methylsulfanyl)phenyl]methyl}-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-ethyl-5-(2-methoxyacetamido)-N-[(2-methoxyphenyl)methyl]-2-(pyridin-3-yl)-1H-1,3-benzodiazole-7-carboxamide
N-({8-[(2-fluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-(phenylsulfanyl)acetamide
1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-{1-[({[1-(morpholin-4-yl)cyclohexyl]methyl}carbamoyl)methyl]-1H-pyrazol-4-yl}-2-(phenylsulfanyl)acetamide
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[2-(1H-imidazol-1-yl)ethyl]piperidin-4-amine
N5-(3-fluorophenyl)-N3,N3-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3,5-dicarboxamide
2-{4-[2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]morpholin-3-yl}acetic acid
2-hydroxy-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide