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(2S,4R)-N-ethyl-4-(4-fluorobenzamido)-1-(1H-pyrrole-3-carbonyl)pyrrolidine-2-carboxamide
methyl 3-({2-[(prop-2-en-1-yl)amino]phenyl}formamido)propanoate
N-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-2-[4-(9H-purin-6-yl)-1H-pyrazol-1-yl]acetamide
(4S)-3-{[4-(difluoromethoxy)phenyl]methyl}-4-(propan-2-yl)-1,3-oxazolidin-2-one
2-[4-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-N-(2-fluorophenyl)-2-oxoacetamide
N-[(3,5-dimethoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)-4-methylpyrimidine-5-carboxamide
2-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-N,N,5-trimethylpyrimidin-4-amine
4-[(4-fluorophenyl)methyl]-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1,4-diazepan-5-one
N-{[3-methyl-7-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
1-[1-(4-{imidazo[1,2-b]pyridazin-3-yl}phenyl)ethyl]piperidine
2-[(3-ethyl-1,2-oxazol-5-yl)methyl]-5-[methyl(2-phenylethyl)amino]-2,3-dihydropyridazin-3-one
(1R,5R)-6-(cyclobutylmethyl)-3-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
1-[2-({[(5-phenyl-1H-pyrazol-3-yl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
methyl 3-acetamido-1-ethyl-5-{[(4-methoxyphenyl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-cyclopentyl-6-oxo-N-[2-(propan-2-yloxy)ethyl]piperidine-3-carboxamide
3-chloro-N-(1-hydroxybutan-2-yl)-5-methoxy-N-[(5-methylthiophen-2-yl)methyl]benzamide
N-[(1-benzylpyrrolidin-3-yl)methyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
N-methyl-N-(1H-pyrazol-5-ylmethyl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
4-(1-{4-[2-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy)ethyl]piperazin-1-yl}-1-oxopropan-2-yl)-1,2-dihydrophthalazin-1-one
1-{[1-(3,4-difluorophenyl)-1H-1,2,4-triazol-5-yl]methyl}-4-phenylpyrrolidin-2-one
N-methyl-2-(5-methyl-1H-pyrazol-1-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
N-(2-fluoro-4-methylphenyl)-2-[(2-propylpyridin-4-yl)formamido]propanamide
2-(1-{[4-(pyridin-3-yl)phenyl]methyl}piperidin-2-yl)pyridine
N-{5H,6H,7H,8H,9H,10H-cyclohepta[b]indol-2-ylmethyl}-3-(6-oxo-1,6-dihydropyridazin-3-yl)propanamide
2-({[1-(2-methoxyphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)-5-methyl-1,3,4-oxadiazole
(1R,3S)-7-(7-fluoro-2-methylquinoline-4-carbonyl)-7-azaspiro[3.5]nonane-1,3-diol
(4aS,7aR)-4-[(dimethylcarbamoyl)methyl]-6,6-dioxo-N-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-({7-[2-(2-chlorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-phenoxypropanamide
2-{4-[1-(6-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]piperazin-1-yl}-1-(pyrrolidin-1-yl)ethan-1-one
4-fluoro-N-{2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]ethyl}benzamide
ethyl 5-{[(2-oxo-1-phenylpyrrolidin-3-yl)formamido]methyl}furan-2-carboxylate
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1H-pyrazol-5-ylmethyl)amine
2-(1-methyl-1H-pyrrol-3-yl)-N-{[8-(3-phenylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
{3-[(4-fluorophenyl)methyl]-1-(2-methylbenzoyl)piperidin-3-yl}methanol
5-cyclopropyl-4-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-1-methyl-1H-pyrazole
3-(pentan-2-yl)-8-[(2-propylpyrimidin-5-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-{[(1,1-dioxo-1λ6-thiolan-3-yl)(ethyl)amino]methyl}-N-(1,3-thiazol-2-yl)benzamide
4-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]-5-(4-fluorophenyl)-2-methylpyrimidine
{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}({[5-(methoxymethyl)furan-2-yl]methyl})amine
1-[(2-chloro-4-fluorophenyl)methyl]-N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
N-[(2-fluorophenyl)methyl]-4-(4-{[2-(thiophen-2-yl)ethyl]amino}piperidin-1-yl)benzamide
3-{5-[2-(morpholin-4-yl)ethyl]-1,3,4-thiadiazol-2-yl}-1-[1-(pyrazin-2-yl)propan-2-yl]urea
N-ethyl-N-{[3-(prop-2-en-1-yloxy)phenyl]methyl}-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
N-[(3S,4R)-1-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)sulfonyl]-4-propylpyrrolidin-3-yl]acetamide
3-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-methyl-1-[4-(1H-1,2,4-triazol-1-yl)phenyl]urea
N-(1-hydroxybutan-2-yl)-2-(pyridin-4-yl)-N-(thiophen-2-ylmethyl)acetamide
methyl 1-ethoxy-2-oxo-8-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
5-(2-methoxyacetamido)-N-[(2-methoxyphenyl)methyl]-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
3-{[3-(3-methylphenoxy)azetidin-1-yl]methyl}pyridine
6-methyl-2-oxo-5-[4-(2-phenylethyl)piperidine-1-carbonyl]-1,2-dihydropyridine-3-carbonitrile