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5-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-3-(2-methylpropyl)-1-(propan-2-yl)-1H-1,2,4-triazole
N-[(3S,4R)-4-(propan-2-yl)-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidin-3-yl]methanesulfonamide
2-(azepan-1-yl)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methylacetamide
N-(3,4-difluorophenyl)-6-[1-(morpholin-4-yl)cyclohexanecarbonyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-phenylprop-2-ynamide
5-[1-(4-methoxybenzoyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
(2E)-1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-3-(pyridin-3-yl)prop-2-en-1-one
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1-(propan-2-yl)piperidin-4-amine
2-{4-[(1-methyl-1H-indol-3-yl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
N-[(3-chlorophenyl)methyl]-1-(1-cyclopropanecarbonylpiperidin-4-yl)piperidine-3-carboxamide
2-methyl-7-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
5-[(2-fluoro-4-methoxyphenyl)methyl]-5-[3-(2-methylpiperidin-1-yl)-3-oxopropyl]pyrrolidin-2-one
5-(1-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1H-1,2,3-triazol-4-yl)pyrimidine
2-(dimethylamino)-7-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-({1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)thiophene-3-carboxamide
1-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-3-[4-(3-methylphenyl)piperazin-1-yl]propan-1-one
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(1H-pyrazol-1-yl)butanamide
2-{4-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]phenyl}-5-methyl-1,3,4-oxadiazole
N-{[2-(2,2-diphenylethyl)-6-oxo-1,6-dihydropyrimidin-4-yl]methyl}acetamide
1-(3,5-dimethylphenyl)-4-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]piperazin-2-one
(2S,4S)-4-amino-N-ethyl-1-[4-(1-phenyl-1H-imidazol-4-yl)benzoyl]pyrrolidine-2-carboxamide
N-[4-(aminomethyl)phenyl]-3-(2-methylphenoxymethyl)piperidine-1-carboxamide
1-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-2-(morpholin-3-yl)ethan-1-one
2-(pyridin-2-ylmethyl)-9-[2-(1H-1,2,4-triazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(2,4-dichloro-6-methylphenyl)methyl]-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
N-[3-(1H-1,3-benzodiazol-2-yl)propyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-[(1-cyclohexylpiperidin-3-yl)methyl]-N-(pyridin-3-ylmethyl)-1H-indazole-3-carboxamide
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[3-(2-chlorophenyl)pyrrolidin-1-yl]ethan-1-one
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
1-(4-cyclopentyl-1,4-diazepan-1-yl)-2-[4-(dimethylamino)phenyl]ethan-1-one
3-({2-[1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
4-[1-benzyl-5-(2,2-diethylcyclopropanecarbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperazin-2-one
5-ethyl-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-(4-{[3-(pyrrolidine-1-carbonyl)-1,2-oxazol-5-yl]methoxy}phenyl)ethan-1-one
methyl (2R,4S)-4-hydroxy-1-[2-(1H-pyrazol-1-yl)benzoyl]piperidine-2-carboxylate
3-(1H-indol-3-yl)-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]propanamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)butanamide
1-(4-{[2-(1H-pyrazol-1-yl)ethyl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
2-(5-acetylthiophen-3-yl)-N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
2-[3-(dimethylamino)propyl]-9-(1H-indol-5-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(2,4-dichlorophenoxy)acetyl]piperazine-2-carboxylic acid
2-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-4-amine
5-[(2-chlorophenyl)methyl]-5-{1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
1-[2-(3-fluorophenyl)ethyl]-5-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]piperidin-2-one
N-ethyl-5-(1-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1H-imidazol-2-yl)pyrimidin-2-amine
1-[(4-fluorophenyl)methyl]-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-[4-(2-methoxyethyl)piperazine-1-carbonyl]-1-[2-(pyridin-2-yl)ethyl]piperidin-2-one
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-[(1-ethyl-1H-imidazol-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane