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5-(hydroxymethyl)-2-methyl-4-({[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]amino}methyl)pyridin-3-ol
5-cyclopropyl-4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-3-methyl-1H-pyrazole
1-{2-[(5-chloropyridin-2-yl)oxy]hex-5-en-1-yl}-4-methyl-1,4-diazepane
4-[(propan-2-yl)amino]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
2-(1H-1,3-benzodiazol-1-yl)-N-[(2,6-dimethoxyphenyl)methyl]propanamide
N-{1-[7-(3-methylbut-2-en-1-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-3-phenylpropanamide
methyl 4-(2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamido)butanoate
4-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-1,4-oxazepan-6-ol
N3-tert-butyl-1-cyclohexyl-N5-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-(cyclopropylmethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylic acid
2-(3-chloro-4-methoxyphenyl)-2-{methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}acetic acid
3-butyl-4-[3-(4-hydroxyphenyl)benzoyl]-1-methylpiperazin-2-one
3-(3,4-dimethoxyphenyl)-N-{[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[3-benzyl-3-(hydroxymethyl)piperidin-1-yl]ethan-1-one
9-[2-(morpholin-3-yl)acetyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(2,3-difluorophenyl)methyl]-3-[4-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
3-{[(1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
2-(4-methyl-1,4-diazepan-1-yl)-N-[2-(6-oxo-3-phenyl-1,4,5,6-tetrahydropyridazin-1-yl)ethyl]acetamide
(3S,5S)-5-(cyclopropylcarbamoyl)-1-{[2-(furan-2-yl)phenyl]methyl}piperidine-3-carboxylic acid
(1S,5R)-3-(2-amino-9H-purin-6-yl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
N-cyclopentyl-N-[(2,5-dimethoxyphenyl)methyl]-2-(5-oxopyrrolidin-2-yl)acetamide
(1-{[1-(1,3-benzothiazole-2-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
(3S,4R)-4-(3-methoxyphenyl)-1-(1-methyl-1H-pyrazole-4-carbonyl)pyrrolidine-3-carboxylic acid
1-(7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(thiophen-2-yl)ethan-1-one
1-{1-[(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)methyl]-3,5-dimethyl-1H-pyrazol-4-yl}ethan-1-one
N-{[7-chloro-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)oxolane-2-carboxamide
9-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
1-[2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]piperidine-3-carboxamide
(1R,7S)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-[(3-methylphenyl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-[5-(thiophen-2-yl)furan-2-yl]propan-1-one
4-methyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)-1,3-oxazole-5-carboxamide
(3R,4R)-1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-cyclopropyl-3-methylpiperidin-4-ol
1-(2-methoxyethyl)-3-methyl-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-ethyl-N-({7-[2-(2-methoxyphenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1-methyl-1H-pyrazole-5-carboxamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-({[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenol
3-(2-ethyl-1H-imidazol-1-yl)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
3-methoxy-N-(1-{7-[(2-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
N-[(2-chlorophenyl)methyl]-5-methanesulfonyl-N-methyl-4-(piperidin-3-yl)pyrimidin-2-amine
3-[(cycloheptylamino)methyl]-1-(2,2-dimethylpropyl)-3-hydroxypiperidin-2-one
4-{3-[(2S)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]piperidin-1-yl}-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
3-{5-[(2S)-4,4-difluoropyrrolidine-2-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
3-{4-[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
(1R,2R,6S,7S)-N-(2-chloro-4-fluorophenyl)-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
(benzylsulfamoyl)(methyl)[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amine
5-(3-chlorothiophene-2-carbonyl)-1-methyl-N-[3-(morpholin-4-yl)propyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
N-{[2-(4-acetylpiperazin-1-yl)-7-methylquinolin-3-yl]methyl}-N-cyclopropyl-3,5-dimethoxybenzamide
3-{2-[(2-hydroxyethyl)({[4-(methylsulfanyl)phenyl]methyl})amino]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one