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(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-ethyl-3-{1-[2-(quinazolin-4-yloxy)acetyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-6-(piperidin-4-yl)pyrimidin-4-amine
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]-3-methylthiophene-2-carboxamide
2-(dimethylamino)-8-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
N-cycloheptyl-2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-(cyclopropylmethyl)-1-(2,6-dimethoxypyridine-3-carbonyl)piperidine-3-carboxylic acid
1,3-dimethyl-6-{4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(1-methoxypropan-2-yl)-3-(6-methylpyridin-3-yl)-1-{[4-(methylsulfanyl)phenyl]methyl}urea
(4aR,8aR)-7-[3-(benzyloxy)propyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
(1S,5R)-6-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-cyclopropyl-N-[(3-methylthiophen-2-yl)methyl]-2,1-benzoxazole-3-carboxamide
N-(1-methylpiperidin-4-yl)-2-(oxolan-2-ylmethoxy)-N-(2-phenylethyl)acetamide
{[4-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-2-yl)phenyl]methyl}dimethylamine
methyl 2-(7-chloro-3-{[methyl(2-phenylethyl)amino]methyl}-2-oxo-1,2-dihydroquinolin-1-yl)acetate
8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
(3aR,6aS)-N-(2-chloro-6-methylphenyl)-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
2-benzyl-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1,3-thiazole-4-carboxamide
N-cyclohexyl-6-fluoro-2-oxo-N-(pyridin-4-ylmethyl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-{[5-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
1-[(2,5-dichlorophenyl)methyl]-3-(dimethyl-1H-1,2,4-triazol-3-yl)urea
1,3-dimethyl-5-{octahydro-1H-pyrido[1,2-a]piperazin-2-yl}-1H-pyrazolo[3,4-d][1,3]thiazole
[4-({[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)phenyl]methanol
3-{1-cyclopentyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenol
4-{2-cyclohexyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-(1-propylpiperidin-4-yl)piperidine
[(2-chlorophenyl)methyl](methyl)(oxan-2-ylmethyl)amine
N-[(2-amino-1,3-thiazol-4-yl)methyl]-3,5-dimethyl-1H-indole-2-carboxamide
5-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-2-phenyl-1H-imidazole-4-carboxamide
5-(2,6-dimethoxy-4-methylphenyl)-N,N-diethylfuran-2-carboxamide
3-[(4-methoxypyridin-2-yl)methyl]-5-(piperidin-4-yl)-5-propylimidazolidine-2,4-dione
5-(4-fluoro-3-methoxyphenyl)-1-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-phenyl-1H-imidazole
2-butyl-N-(3-cyanophenyl)-4-methyl-3-oxopiperazine-1-carboxamide
N-cyclohexyl-3-{[4-(propan-2-yl)pyrimidin-2-yl]amino}propanamide
6-fluoro-N-(1-methylpiperidin-4-yl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
3,5-dimethyl-4-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}pyrrolidin-2-yl)-1,2-oxazole
{[6-(2-methoxyquinolin-3-yl)pyridin-3-yl]methyl}dimethylamine
1-[6-(4-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4-(propan-2-yl)piperazine
N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
3,5-dichloro-N-[(4-methanesulfonylmorpholin-2-yl)methyl]-4-methylbenzamide
butyl 2-benzyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxylate
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-3-[(3-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-[(3R,4R)-3-hydroxy-1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-4-yl]pyridine-2-carboxamide
N'-({1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]pyrrolidin-3-yl}methyl)ethanediamide
1-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(2-methylpropyl)-N-propyl-1H-pyrazole-5-carboxamide
N-{2-[2-(methylsulfanyl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}-4-(trifluoromethyl)benzamide
2-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-yl]quinoxaline
1-cyclopentyl-4-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperazin-2-one
methyl 1-methoxy-2-oxo-8-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylate