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2-ethyl-N-({3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]butanamide
4-[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidine-1-carbonyl]-1,2-dihydrophthalazin-1-one
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[1-(pyridin-4-yl)propan-2-yl]acetamide
2-{6-oxo-7-propyl-2,7-diazaspiro[4.5]decan-2-yl}-N-(pyridin-2-ylmethyl)acetamide
8-chloro-2-{[4-(oxan-4-yl)piperazin-1-yl]methyl}quinoline
1-(2-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-2-oxoethyl)-4-ethylpiperazine-2,3-dione
4-{[2-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}benzonitrile
5-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-amine
2-{[4-(4-methylphenyl)-5-(pyridin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
[(3R,4R)-1-[2-amino-6-(methylamino)pyrimidin-4-yl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
4-(4-fluorophenoxy)-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidine
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-(quinazolin-4-yloxy)ethan-1-one
4-[(2-fluorophenyl)methyl]-3-{2-[4-(2-hydroxyethyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
3-methyl-4-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
7-(2-methylphenyl)-4-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(2,3-dihydro-1H-inden-4-yl)-3-[(2-hydroxypropyl)sulfamoyl]benzamide
2-[(3-methoxyphenyl)methyl]-4-(5-methylthiophene-2-carbonyl)morpholine
6-[(diethylamino)methyl]-N-[1-(furan-2-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
(1S,5R)-3-cyclobutanecarbonyl-6-(4-methylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-3,5-dimethylfuran-2-carboxamide
1-(4-aminopiperidin-1-yl)-2-[(4-methylphenyl)amino]-2-phenylpropan-1-one
2-(hydroxymethyl)-N-(6-methyl-2H-1,3-benzodioxol-5-yl)piperidine-1-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
3-({2-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)-2-(furan-2-ylmethyl)propan-1-ol
methyl(oxan-2-ylmethyl){[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
5-(2-{4-[3-(4-fluorophenyl)-1H-pyrazol-4-yl]-1H-1,2,3-triazol-1-yl}ethyl)-1,3,4-thiadiazol-2-amine
8-methoxy-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
5-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-2-amine
2,6-dimethoxy-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]benzamide
2-{1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1H-1,2,3-triazol-4-yl}benzoic acid
2-(2-{[(4,6-dimethylpyridin-3-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
4-(4-cyclopentylpiperazine-1-carbonyl)-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
N-methyl-N-{[5-({3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonan-7-yl}methyl)furan-2-yl]methyl}methanesulfonamide
N-methyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]acetamide
6-tert-butyl-4-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-1-methyl-1H-pyrazolo[3,4-d]pyrimidine
{2-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]-8-methylquinolin-3-yl}methanol
1-(carbamoylmethyl)-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}piperidine-3-carboxamide
3-(2-carboxyphenyl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-methyl-N-(propan-2-yl)-1-benzofuran-7-carboxamide
{[4-({1-[3-(4-fluorophenyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}(methyl)(quinolin-6-ylmethyl)amine
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-3-(1-methylpiperidin-3-yl)propan-1-one
2-{5-[(1R,2R)-2-phenylcyclopropyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N,5-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(3S,5R)-1-(oxan-4-yl)-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
(2E)-N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-3-(2-chlorophenyl)prop-2-enamide
7-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one