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3-amino-N-[1-(benzenesulfonyl)piperidin-4-yl]-1H-1,2,4-triazole-5-carboxamide
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-2,4-dimethoxy-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
(2S)-2-(methoxymethyl)-N-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)pyrrolidine-1-carboxamide
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-4-(1H-1,2,4-triazol-3-yl)benzamide
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-1-(propan-2-yl)pyrrolidine-3-carboxamide
N-[(3S,4R)-4-hydroxyoxolan-3-yl]-2-(4-methoxyphenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
N-[(4-sulfamoylphenyl)methyl]-2,3-dihydro-1-benzofuran-2-carboxamide
1-(5-{[(5-chloropyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
1-{2-[2-(dimethylamino)ethyl]morpholin-4-yl}-3-(methylsulfanyl)propan-1-one
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-1-(pyrimidin-2-yl)piperidin-4-amine
4-{5-[3-(1H-pyrazol-1-yl)phenyl]-1,2,4-oxadiazol-3-yl}pyridine
N-(1-{1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-4-yl}-2-phenylethyl)-N-methylthiophene-3-carboxamide
3-(3,5-dimethylphenyl)-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}propanamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl]methanol
2-(4-{5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenyl)-2-methylpropanenitrile
2-(1H-pyrazol-1-yl)-N-[3-(pyridin-2-yl)propyl]butanamide
3-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}-1-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]urea
3-(2,5-dioxoimidazolidin-4-yl)-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}propanamide
N-[2-(dimethylamino)pentyl]-2,2,6,6-tetramethylpiperidin-4-amine
({1-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)urea
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}[1-(dimethyl-1,3-thiazol-4-yl)ethyl]methylamine
N-methyl-2-{3-oxo-1-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]piperazin-2-yl}acetamide
1-[4-({1-[(4-methoxypyridin-2-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)piperazin-1-yl]ethan-1-one
3-[1-(3-chloro-4-fluorobenzenesulfonyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
N-[1-(3,4-dimethoxyphenyl)propyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
(2S)-2-amino-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-(1H-imidazol-4-yl)propanamide
4-[4-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]-2-(trifluoromethyl)morpholine
(5S)-5-[({[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]pyrrolidin-2-one
4-(1H-1,2,4-triazol-1-yl)-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}butan-1-one
[(3R,4R)-1-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
1-(2-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}-2-oxoethyl)-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
1-{[3-(1H-pyrazol-3-yl)phenyl]methyl}piperazine
5-methoxy-N-methyl-N-(quinolin-5-ylmethyl)pyrimidin-2-amine
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
2-[2-(3-hydroxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-5,6-dimethylpyridine-3-carbonitrile
2-methyl-4-(4-{[methyl(oxan-2-ylmethyl)amino]methyl}phenyl)butan-2-ol
1-(7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-4-methylpentan-1-one
2-(3-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}propyl)-5-(4-fluorophenyl)-2H-1,2,3,4-tetrazole
8-(2-ethoxyacetyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl (2S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-[3-(4-fluorophenyl)benzamido]pyrrolidine-2-carboxylate
8-(3-fluoropyridin-2-yl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(pyridin-3-ylmethyl)-1H-pyrazol-5-yl]pyrrolidine-1-carboxamide
3-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-6,7-dimethoxy-3,4-dihydroquinazolin-4-one
1-{4-[2-cyclobutyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
3-{2-[4-(2-methylphenoxy)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
N-[(3R,4S)-4-cyclopropyl-1-(3-phenylpropyl)pyrrolidin-3-yl]oxane-4-carboxamide
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-[4-methyl-5-(prop-2-en-1-ylsulfanyl)-4H-1,2,4-triazol-3-yl]piperidine
(3aS,6aR)-3-[2-(pyridin-2-yl)ethyl]-5-(1,3-thiazol-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]pyridine-3-carboxylic acid
8-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]-1-methyl-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione