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N-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-2-(1H-pyrazol-1-yl)butanamide
1-(2-{2-[2-(2-methoxyethyl)-2H-1,2,3,4-tetrazol-5-yl]morpholin-4-yl}-2-oxoethyl)-4,4-dimethylpyrrolidin-2-one
1-benzyl-4-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-pyrazole
N-{[(2R)-1-ethylpyrrolidin-2-yl]methyl}-6-(2-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-[(5-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-1,2,4-oxadiazol-3-yl)methyl]morpholine
4-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
2-ethyl-N-(3-fluorophenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
4-(2,5-dimethylthiophen-3-yl)-2-[5-(methoxymethyl)-4-(2-methylpiperidine-1-carbonyl)-1H-pyrazol-1-yl]pyrimidine
2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-4-methyl-3,4-dihydro-2H-1,4-benzoxazine
ethyl 3-[(3-chlorophenyl)methyl]-1-(2-methoxyacetyl)piperidine-3-carboxylate
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}isoquinoline
2-(3-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-ylmethyl}phenoxy)acetamide
(2S,4R)-N,N-diethyl-1-(2-methylpropanoyl)-4-(3-methylthiophene-2-amido)pyrrolidine-2-carboxamide
1-{2-[4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(4aS,7aR)-1-(3,5-difluoropyridine-2-carbonyl)-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-6-methoxypyrimidin-4-amine
3-methyl-1-[2-(piperidin-1-ylmethyl)phenyl]urea
2-(3,5-difluorophenyl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)acetamide
1-methyl-3-(2-methylpropyl)-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-5-carboxamide
N-[(4-chlorophenyl)methyl]-2-(2-methoxyacetyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-3-(2-fluorophenyl)pyrrolidine
N-[(3R,4S)-1-(furan-2-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3-methanesulfonamidopropanamide
N1-[2-chloro-5-(2-methoxyacetamido)phenyl]-N3-methylpyrrolidine-1,3-dicarboxamide
3-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)pyridin-2-amine
4-(dimethylamino)-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}butanamide
2-tert-butyl-5-[4-(oxolan-2-ylmethyl)piperazine-1-carbonyl]pyrimidin-4-ol
3-(pentan-2-yl)-8-(4-propyl-1,2,3-thiadiazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(4-chloro-2-methoxyphenoxymethyl)-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1,2-oxazole-3-carboxamide
1-[(3-methylphenyl)methyl]-4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidine
N-{3-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-3-oxopropyl}methanesulfonamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-1-cyclopentylpiperidine-3-carboxamide
1-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]-4-(thian-4-yl)piperazine
6-(azepane-1-carbonyl)-5-methyl-N-[(6-methylpyridin-2-yl)methyl]thieno[2,3-d]pyrimidin-4-amine
1-cyclopropyl-N-[2-(3,4-dimethoxyphenyl)propan-2-yl]-6-oxopiperidine-3-carboxamide
2-{4-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]piperidin-1-yl}-7-methoxy-4-methylquinazoline
7-fluoro-3-[2-methoxy-2-(thiophen-2-yl)ethyl]-3,4-dihydroquinazolin-4-one
N-[1-(8-fluoroquinoline-2-carbonyl)piperidin-4-yl]methanesulfonamide
3-[(4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)formamido]-N-(4-fluoro-3-methylphenyl)propanamide
2-[(4-chlorophenyl)methyl]-8-(pyrrolidine-1-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2-(5-methyl-1,2-oxazol-3-yl)piperidine
5-[(3-fluorophenyl)methyl]-7-({[2-(1H-imidazol-1-yl)ethyl]amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
6-(2,5-dimethylfuran-3-yl)-2-(3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
3-(4-methylphenoxymethyl)-1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperidine
6-[4-(hydroxymethyl)piperidin-1-yl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
4-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
4-({1-azabicyclo[2.2.2]octan-3-yl}amino)pyrimidine-5-carboxylic acid
(3S)-1-{1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]piperidine-4-carbonyl}pyrrolidin-3-ol
(1S,9R)-11-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
2-(2-chloro-4-fluorophenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine