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3-(1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
2-[(1-ethyl-1H-pyrazol-3-yl)methyl]-8-methyl-2,8-diazaspiro[4.5]decan-3-one
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-(pyridine-4-carbonyl)piperidin-4-ol
4-[2-(4-fluorophenyl)-2-hydroxyacetyl]-1-(3-methoxyphenyl)piperazin-2-one
(2S,4S)-4-amino-1-(1,1-dioxo-1λ6-thiane-4-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
9-[(2R)-2-hydroxy-2-phenylacetyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
{[4-(difluoromethoxy)phenyl]methyl}(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-2-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-cyclopentyl-N-{[3-(3-fluorophenyl)-1,2-oxazol-5-yl]methyl}-5-oxopyrrolidine-3-carboxamide
4-(2H-1,3-benzodioxol-5-yl)-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
2-[1-(furan-2-ylmethyl)-4-(2-methyl-1,3-benzoxazole-6-carbonyl)piperazin-2-yl]ethan-1-ol
6-ethyl-2-methyl-N-[(3R)-piperidin-3-yl]quinoline-4-carboxamide
4-[4-(3-propyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]quinazoline
3-(1H-1,3-benzodiazol-1-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}propanamide
(3S,9R)-11-(4-fluorobenzoyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine-4-carbonitrile
(1S,5R)-6-(pyridazine-3-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
ethyl 4-{[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-pyrazole-3-carboxylate
N-[6-methyl-5-(pyridin-4-yl)pyridin-2-yl]propanamide
1-[(3-fluorophenyl)methyl]-4-[(2-methyl-1,3-oxazol-4-yl)methyl]piperazin-2-one
1-cyclohexyl-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
1-{5-[4-(benzyloxy)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
1-{2-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
1-(4-methoxyphenyl)-5-methyl-4-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperazin-2-one
N-(3-ethyladamantan-1-yl)-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
1-(2-ethylpyridine-4-carbonyl)-2-methyl-4-(2-methylphenyl)piperazine
4-{1-[(4-fluorophenyl)methyl]-5-(oxolan-3-ylmethyl)-1H-1,2,4-triazol-3-yl}pyridine
4-(2-methoxyethyl)-11-({[3-(trifluoromethoxy)phenyl]methyl}amino)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-ethyl-5-methyl-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-1H-pyrazole-4-carboxamide
5-{[(isoquinolin-5-ylmethyl)(methyl)amino]methyl}pyrimidin-2-amine
1-ethyl-4-{[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-3-methyl-1H-pyrazole
5-methyl-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]pyrazine-2-carboxamide
N-[1-(4-hydroxyphenyl)propyl]-3-methoxy-2,2-dimethylpropanamide
{1-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-3-propylpiperidin-3-yl}methanol
5-[3-(1H-imidazol-1-yl)propyl]-2-(methoxymethyl)-1,3-benzoxazole
N,N-dimethyl-5-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-[(3-methoxyphenyl)methoxy]-4-[(4-methyl-1H-imidazol-5-yl)methyl]-1-(2-methylpropyl)-1,4-diazepan-2-one
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(dimethyl-1H-1,2,4-triazol-1-yl)ethan-1-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
2-cyclopropyl-9-[2-methyl-3-(1H-pyrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
(1R,2S,6R,7S)-4-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-4-azatricyclo[5.2.2.02,6]undecane
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
(1R,4S)-2-{2-[2-(methylsulfanyl)phenyl]pyridine-3-carbonyl}-2-azabicyclo[2.2.1]heptane
(3S,5S)-1-(3-methylbut-2-en-1-yl)-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[4-(difluoromethoxy)benzoyl]piperidine
3-(2-methyl-1H-imidazol-1-yl)-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
5-(2,4-difluorophenoxymethyl)-N-(2,3-dihydroxypropyl)-1,2-oxazole-3-carboxamide
N-cyclopentyl-1-methyl-5-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N,3-dimethyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carboxamide
methyl (2S,4R)-4-[2-(2,4-dioxo-1,3-diazinan-1-yl)benzamido]-1-methylpyrrolidine-2-carboxylate