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6-[3-(1H-pyrazol-3-yl)phenyl]-2-(pyrrolidin-1-yl)pyrimidin-4-amine
N-[(3S)-1-[1-(propan-2-yl)piperidine-4-carbonyl]pyrrolidin-3-yl]acetamide
2,6-difluoro-4-methoxy-N-[(2-methyl-1,3-thiazol-4-yl)methyl]benzamide
2-[N-(1-methylpiperidin-4-yl)-1-[3-(1H-pyrazol-1-ylmethyl)phenyl]formamido]acetic acid
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(3-methylphenyl)benzamide
5-[4-hydroxy-1-(2-phenylpropyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)-1-benzofuran-2-carboxamide
dimethyl({5-[2-(3-phenylpropyl)morpholine-4-carbonyl]furan-2-yl}methyl)amine
1-amino-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}cyclopropane-1-carboxamide
4-{1-[(4-phenoxyphenyl)methyl]azetidin-3-yl}pyridine
N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-2,5-dimethoxybenzamide
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-2-(1H-pyrazol-1-yl)benzamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-4-methylpyrimidin-2-amine
N-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-1-methyl-N-(pyridin-4-ylmethyl)piperidin-4-amine
N-(1H-1,3-benzodiazol-2-yl)-2-{methyl[1-(1,2-oxazol-3-yl)ethyl]amino}acetamide
ethyl 3-[(3-chlorophenyl)methyl]-1-[3-(pyridin-3-yl)propanoyl]piperidine-3-carboxylate
{1-[2-(1H-imidazol-2-yl)benzoyl]-3-(3-phenylpropyl)piperidin-3-yl}methanol
4-(1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
3-(5-chloro-2-methoxybenzoyl)-1-[3-(methylsulfanyl)propyl]piperidine
N,N-diethyl-4-{1H-[1,2,3]triazolo[4,5-b]pyridin-6-yl}benzene-1-sulfonamide
5-[(furan-2-ylmethyl)(methyl)amino]-1-methyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(2,3-dihydro-1-benzofuran-3-yl)-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
(1S,5R)-3-(pyridin-2-ylmethyl)-6-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-6-[(2,6-dimethoxyphenyl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-cyclopropanecarbonyl-1-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indole
N-[(3-chlorophenyl)methyl]-3-{1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]piperidin-4-yl}propanamide
2,3-dimethyl-7-[3-(prop-2-en-1-yloxy)benzoyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
(2R)-N-[3-(2-ethoxyethoxy)phenyl]-2-methylpiperazine-1-carboxamide
3-(5-methyl-1H-pyrazol-1-yl)-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)propanamide
3-methyl-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine
1-(5-chloropyridin-2-yl)-4-(2,3-difluoro-6-methoxybenzoyl)piperazine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
4-(2,2-dimethyloxane-4-carbonyl)-6-[(3-fluorophenyl)methoxy]-1-(2-phenylethyl)-1,4-diazepan-2-one
1-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1,2-dihydroquinolin-2-one
{1-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-2-phenylethyl}(2-methoxyethyl)(pyridin-2-ylmethyl)amine
[(3R,4R)-1-(5-chloro-2-methylbenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[3-(phenylsulfanyl)propyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-ethoxy-5-(2-{[1-(pyridin-4-yl)propyl]amino}pyrimidin-4-yl)benzoic acid
(3aS,6aS)-2-(dimethylcarbamoyl)-5-(6-ethyl-5-fluoropyrimidin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{[(3-ethoxyphenyl)methyl]({[1-(propan-2-yl)piperidin-4-yl]methyl})amino}ethan-1-ol
6-fluoro-2-({4-[(1-methylpiperidin-4-yl)methyl]piperazin-1-yl}methyl)quinolin-4-ol
1-(1H-imidazol-4-ylmethyl)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-{[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}benzonitrile
N-[2-(2,5-dimethylphenoxy)ethyl]-N,1-dimethyl-1H-1,2,3-benzotriazole-5-carboxamide
N-{[2-methoxy-5-(1H-pyrazol-3-yl)phenyl]methyl}cyclopentanamine
(2H-1,3-benzodioxol-5-ylmethyl)[(4-methyl-1H-imidazol-5-yl)methyl](pyridin-3-ylmethyl)amine
N-(2-{2-[4-(1H-imidazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)pyridine-4-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-oxo-1,6-dihydropyridine-2-carboxamide
4-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]piperazine-2-carboxylic acid
(2R,3R)-1'-(furan-3-ylmethyl)-3-(2-methyl-1H-imidazol-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-1,3-diazinane-2,4-dione