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(2S)-2-[({3-ethoxy-4-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]propanamide
1-(2-methoxyphenyl)-4-{2-[4-(propan-2-yl)morpholin-2-yl]acetyl}piperazin-2-one
2-(thianthren-1-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
7-[2-(4-chloro-1H-pyrazol-1-yl)acetyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(1-methyl-1H-pyrazol-5-yl)-1-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]urea
(3S,9aR)-8-[(2,5-dimethylphenyl)methyl]-3-(1H-indol-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}quinoxaline
(2S)-2-methoxy-2-phenyl-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
2-[1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]pyridine
1-butyl-5-(3-phenoxypropyl)-1H-1,2,4-triazole
4-[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]-7-hydroxy-6-methoxy-1,2,3,4-tetrahydroquinolin-2-one
4-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}thiomorpholine
2-(4-methoxypiperidin-1-yl)-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridine
2-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
4-methyl-5-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrimidine
1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
methyl 2-[({3-[(1,4-dimethyl-1H-pyrazol-5-yl)carbamoyl]phenyl}methyl)(methyl)amino]acetate
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl][(4-fluorophenyl)methyl](oxolan-2-ylmethyl)amine
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-3-(1,2-oxazolidin-2-yl)propanamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
7-(1-benzothiophen-3-yl)-9-methoxy-4-(1H-pyrrol-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1R,5S)-6-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}-6-azabicyclo[3.2.1]octane
1-methyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
4-{1-[1-(furan-2-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
2-(2,3-difluorophenoxymethyl)-N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-1,3-oxazole-4-carboxamide
3-(1H-1,3-benzodiazol-2-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]propan-1-one
1-methyl-3-(2-methylpropyl)-N-(2,2,2-trifluoroethyl)-1H-pyrazole-5-carboxamide
3-amino-1-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propan-1-one
4-(4-methoxy-2-methylphenyl)-3,5-dimethyl-1H-pyrazole
(3S,4R)-N-(2,4-difluorophenyl)-3-acetamido-4-(5-methylfuran-2-yl)pyrrolidine-1-carboxamide
4-{5-fluoro-2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]pyrimidin-4-yl}morpholine
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]propan-1-one
4-[5-(1H-1,3-benzodiazol-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]-2-methoxyphenol
3-{[(5-acetylpyridin-2-yl)amino]methyl}-6-cyclopentyl-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
4-[4-(1-hydroxy-2-phenylethyl)piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
1-[3-(1H-imidazol-2-yl)-2,4,6-trimethylphenyl]ethan-1-one
7-(1,3-benzothiazol-2-yl)-4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{[6-(2,3-dimethylphenyl)pyridin-3-yl]methyl}-4-methylpiperazine
N-(2-propyl-2H-1,2,3-triazol-4-yl)-2-[3-(thiophen-3-yl)-1H-pyrazol-1-yl]acetamide
N-[2-(4-methylpiperidin-1-yl)ethyl]-3-(1,2-oxazinan-2-yl)-N-(propan-2-yl)propanamide
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
(1R,5R)-6-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(3,4-difluorobenzoyl)-7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
(3R,4S)-4-(4-methoxyphenyl)-1-(quinoline-6-carbonyl)pyrrolidin-3-amine
1-(4-fluorophenyl)-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-1,4-diazepane
ethyl 3-benzyl-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidine-3-carboxylate
1-[(3-methoxyphenyl)methyl]-4-[2-(morpholin-4-ylmethyl)propanoyl]piperazin-2-one
4-{1-[(1R,2R)-2-phenylcyclopropanecarbonyl]piperidin-4-yl}pyridine
1-ethyl-4-{[2-(pyridin-4-yl)-1H-imidazol-1-yl]methyl}pyrrolidin-2-one