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1-{[5,8-dimethoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}azetidin-3-ol
1-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-4-(3-phenylpropyl)-1,4-diazepane
4-{[methyl(pyrazin-2-ylmethyl)amino]methyl}-N-(1-methyl-1H-1,3-benzodiazol-5-yl)benzamide
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
2-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-4-methylphenol
methyl 1-(2-methylpropyl)-5-[(oxan-4-yl)amino]-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{1-[(4-fluorophenyl)methyl]-4-[3-(1H-pyrazol-1-yl)propyl]piperazin-2-yl}ethan-1-ol
1-(cyclopropylmethyl)-3-hydroxy-3-({[(6-methylpyridin-2-yl)methyl]amino}methyl)piperidin-2-one
4-hydroxy-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[2-(pyridin-2-yl)ethyl]pyrimidine-5-carboxamide
2-methoxy-3-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrazine
3-cyclopentyl-1-[2-(1H-imidazol-5-yl)ethyl]-5-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-1,2,4-triazole
4-(3-{[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]oxy}benzoyl)morpholine
4,6-dimethyl-2-{3-oxa-9-azaspiro[5.5]undecan-9-yl}pyridine-3-carbonitrile
5-(2,6-dimethoxyphenyl)-1-phenyl-1H,4H-pyrazolo[3,4-d]imidazole
1-(2-methylphenyl)-4-[2-(2,3,4-trifluorophenyl)acetyl]piperazin-2-one
1-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-3-ol
2-amino-3-ethyl-N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-[2-oxo-5-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetamide
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
(3R,4R)-1-(3,4-dimethoxybenzenesulfonyl)-3,4-dimethylpyrrolidin-3-ol
1-[(2-chlorophenyl)methyl]-N-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
5-methyl-N-[(6-methylpyridin-2-yl)methyl]-4-{[1-(thiophen-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
5-[5-(trifluoromethyl)pyridin-2-yl]-1,2,3,4-tetrahydroisoquinoline
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
1-ethyl-1-(oxan-4-yl)-3-[2-(propylsulfanyl)phenyl]urea
3-[(3R,4S)-1-[2-(2-methoxyphenyl)acetyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-[(2-chloropyridin-3-yl)methyl]-N,2,7-trimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
[({1-[(2-chloro-4,5-dimethoxyphenyl)methyl]piperidin-3-yl}methyl)sulfamoyl]dimethylamine
1-methyl-3-(2-methylpropyl)-N-[3-oxo-3-(pyrrolidin-1-yl)propyl]-1H-pyrazole-5-carboxamide
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]-1,2,5-thiadiazole-3-carboxamide
5-[(benzyloxy)methyl]-3-(oxolan-3-yl)-1H-1,2,4-triazole
5-cyclobutanecarbonyl-3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
4-(1-methyl-1H-1,2,4-triazol-5-yl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]pyrimidin-2-amine
3,5,7-trimethyl-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)-1H-indole-2-carboxamide
5-(2-fluorophenyl)-N-methyl-N-(pyrazin-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrazolo[1,5-a]pyridine-3-carboxamide
(1S,9S)-11-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
1-(4,6-dimethylpyrimidin-2-yl)-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}piperidin-4-amine
N-[(4-fluorophenyl)methyl]-4,6-dimethyl-2-oxo-N-(oxolan-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
[1-(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methanamine
methyl 4-[2-amino-3-cyano-6-(4-hydroxy-2-methylphenyl)pyridin-4-yl]-1H-pyrazole-3-carboxylate
5-(6-chloropyridin-2-yl)-N-[2-(dimethylamino)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-methyl-N-[1-(pyridin-3-yl)propyl]-4-sulfamoylbenzamide
2-({[(1-methyl-1H-pyrazol-4-yl)methyl](propan-2-yl)amino}methyl)benzoic acid
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}({2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl})amine
2-(dimethylamino)-2-(3-fluorophenyl)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)acetamide
1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-(dimethylamino)-2-(2-methylphenyl)ethan-1-one
1-benzyl-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-(2-methoxyethyl)-2-(6-methoxynaphthalen-2-yl)morpholine