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N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
5-methoxy-1,2-dimethyl-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
N-[(4-fluorophenyl)methyl]-3-{1-[2-(pyridin-2-yl)acetyl]piperidin-4-yl}propanamide
ethyl 5-{[(1-hydroxypropan-2-yl)amino]methyl}-1-(4-phenyl-1,3-thiazol-2-yl)-1H-pyrazole-4-carboxylate
N-[(5-methylpyrazin-2-yl)methyl]-2-oxo-1-phenylpyrrolidine-3-carboxamide
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propan-1-one
1-[(2-{[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]oxy}phenyl)methyl]-4-methylpiperazine
N-methyl-2-[5-oxo-3-phenyl-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
2-(3-{[3-(3-methoxyphenoxy)azetidin-1-yl]methyl}phenoxymethyl)pyridine
2-(dimethylamino)-8-[(2-ethylpyrimidin-4-yl)methyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-[3-(cyclohexyloxy)propyl]-4-methylpyrimidin-2-amine
2-{[6-(methoxymethyl)pyridin-2-yl]formamido}-N-(propan-2-yl)acetamide
3-{4-[1-(4-fluorophenyl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}-1λ6-thiolane-1,1-dione
4-(4-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidin-2-amine
[(1-ethyl-1H-pyrazol-4-yl)methyl][1-(4-methylphenyl)propan-2-yl]amine
1-(2,6-dimethylbenzoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(1s,4s)-4-{4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}cyclohexan-1-amine
(3R,4S)-4-cyclopropyl-N,N-dimethyl-1-[4-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-amine
(2S,4R)-4-amino-1-(2,6-dimethoxybenzoyl)-N-ethylpyrrolidine-2-carboxamide
3-ethyl-1-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)urea
N-cyclopropyl-2-(dimethylamino)-2-(4-fluorophenyl)-N-(1,3-thiazol-2-ylmethyl)acetamide
1-[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-3-ethylpiperazine
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-4-yl]propanamide
(3S,5R)-5-[(4-fluorophenyl)carbamoyl]-1-(2-phenylethyl)piperidine-3-carboxylic acid
2-(2-{1-[(2R)-2-cyclohexyl-2-hydroxyacetyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
1-methyl-5-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(3,4-difluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]propan-1-one
N-[(3R,4R)-1-(5-ethyl-1,2,4-oxadiazol-3-yl)-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
1-[2-(quinolin-4-yloxy)hex-5-en-1-yl]piperidine-4-carboxylic acid
N-(4-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}phenyl)acetamide
N-[2-(oxolan-2-ylmethoxy)phenyl]-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
2-amino-7-(4-phenoxybutanoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
7-(2-hydroxyethyl)-2-(8-methoxyquinolin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[3-(4-methoxyphenoxy)propyl]-N-methyl-2-propanamidopropanamide
3-{5-[(1R,2S,3S,4R,5S)-tricyclo[3.2.1.02,4]octan-3-yl]-1,2,4-oxadiazol-3-yl}pyridazine
2-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]-3,4-dihydroquinazolin-4-one
3-{[2-(dimethylamino)pyridin-3-yl]methyl}-1-(3-fluorophenyl)urea
[1-(5-methyl-1,3-diphenyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]methanol
N-[(3R,4R)-3-hydroxy-1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl]pyridine-3-carboxamide
N-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-1-(2-fluorophenyl)cyclopropane-1-carboxamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[(5-propylfuran-2-yl)methyl]pyrrolidin-3-yl]methanol
5-{4-[4-phenyl-1-(pyridin-3-ylmethyl)-1H-imidazol-5-yl]phenyl}pyrimidine
2-chloro-4-{1-[2-(4-ethylpiperazin-1-yl)-2-methylpropyl]-1H-imidazol-2-yl}phenol
(3R,4R)-3-cyclopropyl-1-(4-methanesulfonylbenzoyl)-4-methylpyrrolidin-3-ol
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
3-(2-chlorophenyl)-1-(4-fluorophenyl)-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1H-pyrazole
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-1-(pyridine-2-carbonyl)piperidine-4-carboxamide
8-(6-cyclopropylpyrimidin-4-yl)-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-N'-(4-methylphenyl)-N-[3-(pyrrolidin-1-yl)propyl]propanediamide
3-[(2-amino-5-ethylpyrimidin-4-yl)(methyl)amino]-1-phenylpropan-1-ol