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2-[5-(quinoxalin-2-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-1,4-diazepan-5-one
2-{7,7-dimethyl-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}-N-(2,4-dimethylphenyl)acetamide
1-ethyl-7-methyl-4-oxo-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,4-dihydro-1,8-naphthyridine-3-carboxamide
3-[5-(2,3-dihydro-1H-indene-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-4-[(2-hydroxyethyl)sulfamoyl]benzamide
5-methoxy-N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)-4-oxo-1,4-dihydropyridine-2-carboxamide
dimethyl({4-methyl-5-[1-(oxan-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-2-(3-hydroxyphenyl)ethan-1-one
1-ethyl-5-(2-methoxyacetamido)-2-(pyridin-3-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-1,3-benzodiazole-7-carboxamide
N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-1-(piperidin-1-yl)cyclohexane-1-carboxamide
6-(dimethylamino)-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]pyridine-3-carboxamide
N-({4-[(3,5-dimethoxyphenyl)methoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-4-(trifluoromethyl)benzamide
1-(1,3-benzothiazol-2-ylmethyl)-3-{1-[2-(dimethylamino)ethyl]-3-methyl-1H-pyrazol-5-yl}-1-methylurea
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(trifluoromethyl)benzamide
3-{4-[4-(1-methoxypropan-2-yl)piperidin-1-yl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
(5-{1-[2-methoxy-1-(pyridin-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}furan-2-yl)methanol
(3S,4R)-1-[6-(dimethylamino)pyridine-3-carbonyl]-4-methylpiperidine-3,4-diol
2,5-dioxo-6-(3,3,3-trifluoro-2-hydroxypropyl)-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
6-methyl-2-[3-({4-[(pyrimidin-2-yl)amino]piperidin-1-yl}methyl)phenyl]-3,4-dihydropyrimidin-4-one
N-(3-hydroxypropyl)-2-methoxy-N-[(5-methylthiophen-2-yl)methyl]pyridine-3-carboxamide
3-{imidazo[1,2-a]pyridin-2-yl}-5-[5-(propan-2-yl)-1,2-oxazol-3-yl]-1,2,4-oxadiazole
2-[(1S,5R)-3-(5-chloro-2-oxo-1,2-dihydropyridine-3-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-(furan-2-ylmethyl)-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(2-methylpropyl)propanamide
3-methyl-8-{1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(butan-2-yl)-2-(3-chloro-4-hydroxyphenyl)-N-cyclopentylacetamide
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(trifluoromethyl)pyrimidin-4-amine
1-[4-(2-methoxyphenyl)piperazin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
(3R,4R)-4-amino-1-{4-[(butylsulfanyl)methyl]-5-methylfuran-2-carbonyl}piperidin-3-ol
2-[4-(2-amino-6-methylpyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-cyclopentyl-1H-pyrazol-5-yl)acetamide
N-[(3-chloro-2-fluorophenyl)methyl]-2,2-dimethyloxane-4-carboxamide
(3S,4R)-1-(2,5-dimethylfuran-3-carbonyl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
1-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-4-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-1,2,3-triazole
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-4-(4-methylphenoxy)piperidine-4-carboxamide
1-(azocan-1-yl)-3-(2-methoxy-5-{[(2-methoxyethyl)amino]methyl}phenoxy)propan-2-ol
2-{N-methyl-1-[4-(piperidin-1-ylmethyl)phenyl]formamido}-2-(pyridin-3-yl)acetic acid
4-[6-(propan-2-yl)pyrimidin-4-yl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(1-methyl-1H-imidazol-2-yl)-1-[4-(5-methylfuran-2-yl)benzoyl]piperidine
2-[1-(propan-2-yl)-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
9-[(5-methylthiophen-2-yl)methyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-methyl-4-phenylpyrimidine-5-carboxamide
6-methyl-2-{[methyl({2-[2-(prop-2-en-1-yl)phenoxy]ethyl})amino]methyl}pyridin-3-ol
2-(4-fluorophenyl)-1-[5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl]azetidine
3-{5-[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]-4-phenyl-1H-imidazol-1-yl}propanamide
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-3-phenyl-1,2,4-oxadiazol-5-amine
3-[(3S)-3-ethylmorpholine-4-carbonyl]-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
N-{1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}pyridin-2-amine
5-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
(4aS,8aR)-1-(3-methoxypropyl)-6-(pyrrolidine-1-carbonyl)-decahydro-1,6-naphthyridin-2-one